Comprehensive heterocyclic chemistry III: [a review of the literature 1995 - 2007] 15 Cumulative subject index
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Format: | Buch |
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Sprache: | English |
Veröffentlicht: |
Amsterdam [u.a.]
Elsevier
2008
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Ausgabe: | 1. ed. |
Online-Zugang: | Inhaltsverzeichnis |
Beschreibung: | LIX, 350 S. Ill. |
ISBN: | 9780080450070 |
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245 | 1 | 0 | |a Comprehensive heterocyclic chemistry III |b [a review of the literature 1995 - 2007] |n 15 |p Cumulative subject index |c execut.-ed. Alan R. Katritzky. Eds-in-chief Christopher A. Ramsden ... |
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700 | 1 | |a Katritzky, Alan R. |d 1928-2014 |e Sonstige |0 (DE-588)137133421 |4 oth | |
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Datensatz im Suchindex
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adam_text | Contents of All Volumes
VOLUME 1 THREE-MEMBERED HETEROCYCLES, TOGETHER WITH
ALL FUSED SYSTEMS CONTAINING A THREE-MEMBERED
HETEROCYCLIG RING
1.01 Aziridines and Azirines: Monocyclic 1
A PADWA, Emory University, Atlanta, GA, USA
1.02 Aziridines and Azirines: Fused-ring Derivatives 105
M C McMILLS and S C BERGMEIER, Ohio University, Athens, OH, USA
1.03 Oxiranes and Oxirenes: Monocyclic 173
G DAKE, University of British Columbia, Vancouver, BC, Canada
1.04 Oxiranes and Oxirenes: Fused-ring Derivatives 235
D M HODGSON, University of Oxford, Oxford, UK
M A H STENT, Key Orgamcs Ltd., Cornwall, UK
1.05 Thiiranes and Thiirenes: Monocyclic 299
J WARKENTIN, McMaster University, Hamilton, ON, Canada
D PLAZUK, University of Lodz, Lodz, Poland
1.06 Thiiranes and Thiirenes: Fused-ring Derivatives 391
T VILAIVAN, W CHAVASIRI, and P RASHATASAKHON, Chulalongkorn University,
Bangkok, Thailand
1.07 Three-membered Rings with One Selenium or Tellurium Atom 433
R S GLASS, The University of Arizona, Tucson, AZ, USA
1.08 Phosphiranes, Phosphirenes, and Heavier Analogues 457
H HEYDT, Technische Universitdt Kaiserslautern, Kaiserslautern, Germany
1.09 Three-membered Rings with One Silicon, Germanium, Tin or Lead Atom 483
M A MENDEZ-ROJAS, Universidadde las Americas, Cholula, Mexico
G MERINO, Universidad de Guanajuato, Guanajuato, Mexico
1.10 Three-membered Rings with One Boron Atom 513
N FARFAN, Universidad National Autonoma de Mexico, Mexico City, Mexico
H I BELTRAN, Universidad Autonoma Metropolitana, Cuajimalpa, Mexico City, Mexico
1.11 Diaziridines and Diazirines 539
G D McALLISTER, A PERRY, and R J K TAYLOR, University of York, York, UK
1.12 Oxaziridines and Oxazirines 559
F A DAVIS, Temple University, Philadelphia, PA, USA
B-C CHEN, Bristol-Myers Squib/? Company, Princeton, NJ, USA
P ZHOU, Wyeth Research, Princeton, NJ, USA
v
vj Contents
1.13 Thiaziridines and Thiazirenes
U ZOLLRR, Haifa University - Oranim, Kiryat Tivon, Israel
1 14 Three-membered Rings with Two Oxygen and/or Sulfur Atoms 641
M ROJE and T PORTADA, Ructer Boskovic Institute, Zagreb, Croatia
1.15 Three-membered Rings with Two Heteroatoms including Selenium or Tellurium;
Three-membered Rings with Three Heteroatoms °79
L NYULASZI and Z BENKO, Budapest University of Technology
and Economics, Budapest, Hungary
1.16 Three-membered Rings with Two Heteroatoms including Phosphorus to Bismuth 695
L WEBER, Unhersitat Bielefeld, Bielefeld, Germany
1.17 Three-membered Rings with Two Heteroatoms including Other Elements 749
T M GILBERT, Northern Illinois University, DeKalb, IL, USA
Index 79-S
VOLUME 2 FOUR-MEMBERED HETEROCYCLES TOGETHER WITH
ALL FUSED SYSTEMS CONTAINING A FOUR-MEMBERED
HETEROCYCLIC RING
2.01 Azetidines, Azetines and Azetes: Monocyclic 1
G S SINGH, University of Botswana, Gaborone, Botswana
M D HOOGHE, Ghent University, Ghent, Belgium
N DE KIMPE, Ghent University, Ghent, Belgium
2.02 Cephalosporins 111
B ALCAIDE and C ARAGONCILLO, Unwersidad Complutense de Madrid, Madrid, Spain
P ALMENDROS, Instituto de Quimica Orgdnica General, CSIC, Madrid, Spain
2.03 Penicillins 173
J MARCHAND-BRYNAERTand C BRULE, Umversite catholtque de Louvain,
l.ouvain-la-Neuve, Belgium
2.04 Other Fused Azetidines, Azetines and Azetes 239
L K MEHTA and J PARRICK, Brunei University, Uxbridge, UK
2.05 Oxetanes and Oxetenes: Monocyclic 321
H C HAILES, University College London, London, UK
J M BEHRENDT, Aston University, Birmingham, UK
2.06 Oxetanes and Oxetenes: Fused-ring Derivatives 365
P H DUSSAULT and C XU, University of Nebraska - Lincoln, Lincoln, NE, USA
2.07 Thietanes and Thietes: Monocyclic 389
S LESNIAK, W J KINART, and J LEWKOWSKI, University of Lodz, Lodz, Poland
2.08 Thietanes and Thietes: Fused-ring Derivatives 429
S LESNIAK, W J KINART, and J LEWKOWSKI, University of Lodz, Lodz, Poland
2.09 Four-membered Rings with One Selenium or Tellurium Atom 463
M KOKKTSU and H ISHIHARA, Gifu University, Gifu, Japan
2.10 Four-membered Rings with One Phosphorus, Arsenic, Antimony, or Bismuth Atom 479
I KAWASHIMA and J KOBAYASHI, The University of Tokyo, Tokyo, Japan
2.11 Four-membered Rings with One Silicon, Germanium, Tin, or Lead Atom 511
M V KOZYTSKA and G B DUDLEY, The Florida State University, Tallahasee, FL, USA
ZM Four-membered Rings with One Boron or Other Atom c55
1 IORITA, R C BAUER, and j M STRYKER, University of Alberta, Edmonton
AB, Canada
i
I
Contents vii
2.13 Four-membered Rings with Two Nitrogen Atoms 623
B B LOHRAY and V B LOHRAY, Bhuvid Research Laboratory, Pvt. Ltd.,
Ahmedabad, India
B K SRIVASTAVA, Zydus Research Center, Ahmedabad, India
2.14 Four-membered Rings with One Oxygen and One Nitrogen Atom 689
S FLORIO, V CAPRIATI, and R LUISI, Universitd di Ban, Ban, Italy
2.15 Four-membered Rings with One Sulfur and One Nitrogen Atom 713
P HUDHOMME, UniversitedAngers, Angers, France
2.16 Four-membered Rings with Two Oxygen Atoms 775
D K TAYLOR, The University of Adelaide, Adelaide, SA, Australia
2.17 Four-membered Rings with One Oxygen and One Sulfur Atom 795
D K TAYLOR, The University of Adelaide, Adelaide, SA, Australia
2.18 Four-membered Rings with Two Sulfur Atoms 811
J DRABOWIQZ, Polish Academy of Sciences, Czestochowa, Poland, Jan Dlugosz University
of Czestochowa, Czestochowa, Poland
J LEWKOWSKI, University of Lodz, Lodz, Poland
W KUDELSKA, Jan Dlugosz University of Czestochowa, Czestochowa, Poland
A ZAJAC, Polish Academy of Sciences, Lodz, Poland
2.19 Four-membered Rings with Two or More Heteroatoms including Selenium
or Tellurium 853
T SHIMIZU, Tokyo Metropolitan University, Tokyo, Japan
2.20 Four-membered Rings with Two Heteroatoms including Phosphorus to Bismuth 875
U ZENNECK and M HOFMANN, University of Erlangen-Nurnberg, Erlangen, Germany
2.21 Four-membered Rings with Two Heteroatoms including Silicon to Lead 907
M CYPRYK, Polish Academy of Sciences, Lodz, Poland
A JOZWIAK, University of Lodz, Lodz, Poland
2.22 Four-membered Rings with Three Heteroatoms with at least One Oxygen,
Sulfur or Nitrogen Atom 939
A SACKUS, Kaunas University of Technology, Kaunas, Lithuania
F A SL0K, Vipergen ApS, Copenhagen, Denmark
2.23 Four-membered Rings with Three Heteroatoms not including Oxygen,
Sulfur or Nitrogen Atom 973
E LUKEVICS and E ABELE, Latvian Institute of Organic Synthesis, Riga, Latvia
Index 991
VOLUME 3 FIVE-MEMBERED RINGS WITH ONE HETEROATOM
TOGETHER WITH THEIR BENZO AND OTHER CARBOCYGLIG-FUSED
DERIVATIVES
3.01 Pyrroles and their Benzo Derivatives: Structure 1
M D ISCHIA, A NAPOLITANO, and A PEZZELLA, University of Naples
Federico II , Naples, Italy
3.02 Pyrroles and their Benzo Derivatives: Reactivity 45
B A TROFIMOV and N A NEDOLYA, Russian Academy of Sciences - Siberian
Branch, Irkutsk, Russia
3.03 Pyrroles and their Benzo Derivatives: Synthesis 269
J BERGMAN and T JANOSIK, Karolinska Institute, Huddinge, Sweden
3.04 Pyrroles and their Benzo Derivatives: Applications 353
M D ISCHIA, A NAPOLITANO and A PEZZELLA, University of Naples Federico II ,
Naples, Italy
vjj! Contents
ion
3.05 Furans and their Benzo Derivatives: Structure Joy
A SKNNING, Technical University of Denmark, Kgs. Lyngby, Denmark
3 06 Furans and their Benzo Derivatives: Reactivity 407
H N C WONG, The Chinese University of Hong Kong, Hong Kong, People s Republic of China
K-S YEUNG, Bristol-Myers Squibb Pharmaceutical Research Institute, Wallingford, CT, USA
Z YANG, Peking University, Beijing, People s Republic of China
3.07 Furans and their Benzo Derivatives: Synthesis 497
T GRAENING and F THRUN, TU Berlin, Berlin, Germany
3.08 Furans and their Benzo Derivatives: Applications 571
B A KEAY and J M HOPKINS, University of Calgary, Calgary, AB, Canada
P W DIBBLE, University of Lethbridge, Lethbridge, AB, Canada
3.09 Thiophenes and their Benzo Derivatives: Structure 625
P MOLINA, A ARQUES, and I CARTAGENA, University of Murcia, Murcia, Spain
3.10 Thiophenes and their Benzo Derivatives: Reactivity 741
S RAJAPPA, B-l, Melody Apartments, ICS Colony, Pune 411007, India
A R DESHMUKH, National Chemical Laboratory, Pune, India
3.11 Thiophenes and their Benzo Derivatives: Synthesis 843
O SATO and J NAKAYAMA, Saitama University, Saitama, Japan
3.12 Thiophenes and their Benzo Derivatives: Applications 931
J SCHATZ, T BRENDGEN, and D SCHUHLE, University of Ulm, Ulm, Germany
3.13 Selenophenes 975
F T PELKEY, Hobart and William Smith Colleges, Geneva, NY, USA
3.14 Tellurophenes 1007
V I MINKIN and I D SADEKOV, Rostov State University, Rostov on Don, Russia
3.15 Phospholes 1029
R REAU, University of Rennes 1, Rennes, France
P W DYER, Durham University, Durham, UK
3.16 Arsoles, Stiboles, and Bismoles U49
V MILATA, Slovak Technical University, Bratislava, Slovakia
3.17 Siloles, Germoles, Stannoles, and Plumboles 1181
B WRACKMEYER and O L TOK, Universitdt Bayreuth, Bayreuth, Germany
3.18 Boroles j 22S
G VARVOUNIS, University of loannina, loannina, Greece
3.19 Five-membered Rings with Other Elements 1243
A P SADIMENKO, University of Fort Hare, Alice, South Africa
lndex 1305
VOLUME 4 FIVE-MEMBERED RINGS WITH TWO HETPROATOMS
EACH WITH THEIR FUSED GARBOCYCLIG DERIVATIVES
4.01 Pyrazoles
L ET, Albany Molecular Research, Inc., Albany, NY, USA
4.02 Imida/oles
N XI, Q HUANG, and L LIU, Amgen, Inc., Thousand Oaks, CA, USA
4.03 Isoxazoles
F MArHiaTX,F /MCORDERO U™ersita di Firenze, Sesto Fiorentmo, Italy ^
r Aim.Ht. i 11, Istituto di chimica dei composti organometallki del CNR Sesto
riorenttno, Italy
Contents ix
4.04 Oxazoles 487
V YEH, Astellas Research Institute of America, Skokie, IL, USA
R IYENGAR, Enanta Pharmaceuticals Inc., Watertown, MA, USA
4.05 Isothiazoles 545
F CLERICI, M L GELMI, and S PELLEGRINO, Universita di Mi/ano, Milan, Italy
4.06 Thiazoles 635
B CHEN and W HEAL, The University of Sheffield, Sheffield, UK
4.07 1,2-Selenazoles 755
J MLOCHOWSKI, Wroclaw University of Technology, Wroclaw, Poland
4.08 1,3-Selenazoles 791
M KOKETSU and H ISHIHARA, Gifu University, Gifu, Japan
4.09 1,2-Dioxoles and 1,2-Oxathioles 823
R A AITKEN and L A POWER, University of St. Andrews, St. Andrews, UK
4.10 1,3-Dioxoles and 1,3-Oxathioles 841
R A AITKEN and L A POWER, University of St. Andrews, St. Andrews, UK
4.11 1,2-DithioIes 893
R MARKOVIC and A RASOVIC, University of Belgrade, Belgrade, Serbia
4.12 1,3-Dithioles 955
P BALGZEWSKI, Centre of Molecular and Macromolecular Studies PAS Lodz, Poland
W KUDELSKA, Jan Dtugosz University (JDU), Cz§stochowa, Poland
A BODZIOGH, Centre of Molecular and Macromolecular Studies PAS Lodz, Poland
4.13 Five-membered Rings with Two Adjacent Heteroatoms with at least One Selenium
or Tellurium 1091
M B NIELSEN, University of Copenhagen, Copenhagen, Denmark
4.14 Five-membered Rings with Two Nonadjacent Heteroatoms with at least One
Selenium or Tellurium 1119
M B NIELSEN, University of Copenhagen, Copenhagen, Denmark
4.15 Five-membered Rings with Two Adjacent Heteroatoms with at least One
Phosphorus, Arsenic, or Antimony 1155
K KARAGHIOSOFF, Ludwig-Maximilians Universitat, Munich, Germany
4.16 Five-membered Rings with Two Nonadjacent Heteroatoms with at least One
Phosphorus, Arsenic, or Antimony 1169
J A JOULE, The University of Manchester, Manchester, UK
4.17 Five-membered Rings with Two Adjacent Heteroatoms with at least One Boron 1189
A J ASHE, III, University of Michigan, Ann Arbor, MI, USA
4.18 Five-membered Rings with Two Nonadjacent Heteroatoms with at least One Boron 1225
G VARVOUNIS, University of Ioannina, loannina, Greece
4.19 Five-membered Rings with Two Adjacent Heteroatoms with at least One
Other Element 1243
C CANO-SOUMILLAC, Northern Institute for Cancer Research, Newcastle-upon-Tyne, UK
4.20 Five-membered Rings with Two Nonadjacent Heteroatoms with at least One
Other Element 1271
C CANO-SOUMILLAC, Northern Institute for Cancer Research, Newcastle-upon-Tyne, UK
Index 1305
x Contents
VOLUME 5 FIVE-MEMBERED RINGS: TRIAZOLES, OXADIAZOLES
THIADIAZOLES AND THEIR FUSED GAJRBOCYCLIC DERIVATIVES
5.01 1,2,3-Triazoles !
S RACHWAL, Cortex Pharmaceuticals, Inc., Irvine, CA, USA
A R KATRITZKY, University of Florida, Gainesville, FL, USA
5.02 1,2,4-Triazoles K
A D M CURTIS and N JENNINGS, Keele University, Keele, UK
5.03 1,2,3-Oxadiazoles 211
VV FRASER, Aston University, Birmingham, UK
5.04 1,2,4-Oxadiazoles 243
K HEMMING, University of Huddersfield, Huddersfield, UK
5.05 1,2,5-Oxadiazoles 315
G NIKONOV and S BOBROV, Alchem Laboratories Co., Alachua, FL, USA
5.06 1,3,4-Oxadiazoles 397
J SUWINSKI and W SZCZEPANKIEWICZ, Silesian University of Technology,
Gliwice, Poland
5.07 1,2,3-Thiadiazoles 467
D J WILKINS, Key Organics Limited, Camelford, UK
5.08 1,2,4-ThiadiazoIes 487
D J WILKINS, Key Organics Limited Camelford, UK
5.09 1,2,5-Thiadiazoles 515
P A KOUTENTIS, University of Cyprus, Nicosia, Cyprus
5.10 1,3,4-Thiadiazoles 567
P A KOUTENTIS, University of Cyprus, Nicosia, Cyprus
C P CONSTANTINIDES, The University of Cambridge, Cambridge, UK
Index 607
VOLUME 6 OTHER FIVE-MEMBERED RINGS WITH THREE OR MORE
HETEROATOMS, AND THEIR FUSED CARBOCYGLIC DERIVATIVES
6.01 l,2-Oxa/thia-3-azoles 1
O A RAKITIN, Zelinski Institute of Organic Chemistry, Moscow, Russia
6.02 l,3-Oxa/thia-2-azoles 37
C) A RAKITIN, Zelinsky Institute of Organic Chemistry, Moscow, Russia
6.03 l,2-Oxa/thia-4-azoles 6J
N N MAKHOVA, Zelinsky Institute of Organic Chemistry, Moscow, Russia
6.04 l,4-Oxa/thia-2-azoles jq5
N G ARGYROPOULOS, Aristotle University ofThessaloniki, Thessaloniki, Greece
6.05 Fiye-membered Rings with Three Oxygen or Sulfur Atoms in 1,2,3-Positions 145
V SAMOSHIN, University of the Pacific, Stockton, CA, USA
6.06 Five-membered Rings with Three Oxygen or Sulfur Atoms in 1,2,4-Positions 191
1 S BALABAN, Karlsruhe Institute of Technology, Karlsruhe, Germany
A 1 BALABAN, Texas A M University at Galveston, Galveston, IX USA
6.07 Tetrazoles
lAf?f ?r ?? V ^OLDOBSKII »d R E TRIFONOV, Si. Petersburg State
Institute of Technology, St. Petersburg, Russia
Contents xi
6.08 Oxatriazoles 425
W FRASER, Aston University, Birmingham, UK
6.09 1,2,3,4-Thiatriazoles 441
W DEHAEN, University of Leuven, Leuven, Belgium
V A BAKULEV, The Urals State Technical University, Ekaterinburg, Russia
6.10 1,2,3,5-Thiatriazoles 485
V A BAKULEV, The Urals State Technical University, Ekaterinburg, Russia
W DEHAEN, University of Leuven, Leuven, Belgium
6.11 1,2,3,5-Dithiadiazoles and 1,3,2,4-Dithiadiazoles 499
R J PEARSON, Keele University, Keele, UK
6.12 Three or Four Heteroatoms including at least One Selenium or Tellurium 517
S YAMAZAKI, Nara University of Education, Nara, Japan
6.13 Three or Four Heteroatoms including at least One Phosphorus 583
V V ZHDANKIN, University of Minnesota Duluth, Duluth, MN, USA
6.14 Three or Four Heteroatoms including at least One Arsenic or Antimony 603
A SCHMIDPETER and K KARAGHIOSOFF, Ludwig-Maximilians-Universitat, Munich,
Germany
6.15 Three or Four Heteroatoms including at least One Boron 615
MVR REDDY, J S CHANDRA, and V J REDDY, University of Minnesota Duluth,
Duluth, MN, USA
6.16 Three or Four Heteroatoms including at least One Silicon 655
T MULLER, Carl von Ossietzky University Oldenburg, Oldenburg, Germany
6.17 Three or Four Heteroatoms including at least One Other Element 691
V N NEMYKIN, University of Minnesota Duluth, Duluth, MN, USA
6.18 Pentazoles 739
T M KLAPOTKE and A HAMMERL, Ludwig-Maximilians Unwersitat Munchen,
Munich, Germany
Index 759
VOLUME 7 SIX-MEMBERED RINGS WITH ONE HETEROATOM, AND THEIR
FUSED GARBOGYCLIC DERIVATIVES
7.01 Pyridines and their Benzo Derivatives: Structure 1
J B HARPER, University of New South Wales, Sydney, NSW, Australia
7.02 Pyridines and their Benzo Derivatives: Reactivity at the Ring 41
D L COMINS, North Carolina State University, Raleigh, NC, USA
S O CONNOR, Clemson University, Clemson, SC, USA
R S AL-AWAR, Eli Lilly and Company, Indianapolis, IN, USA
7.03 Pyridines and their Benzo Derivatives: Reactivity of Substituents 101
V CAPRIO, University of Auckland, Auckland, New Zealand
7.04 Pyridines and their Benzo Derivatives: Reactivity of Reduced Compounds 171
D BARKER, The University of Auckland, Auckland, New Zealand
7.05 Pyridines and their Benzo Derivatives: Synthesis 217
P A KELLER, University ofWollongong, Wollongong, NSW, Australia
7.06 Pyridines and their Benzo Derivatives: Applications 309
C H MCATEER, Vertellus Specialties Inc., Indianapolis, IN, USA
M BALASUBRAMANIAN, Pfizer Inc., Groton, CT, USA
R MURUGAN, Vertellus Specialties Inc., Indianapolis, IN, USA
xjj Contents
7 07 Pyrans and their Benzo Derivatives: Structure and Reactivity 337
A J PHILLIPS, J A HENDERSON, and K L JACKSON, University of Colorado,
Boulder, CO, USA
7 08 Pyrans and their Benzo Derivatives: Synthesis
M A BRIMBLE, J S GIBSON, and J SPERRY, The University of Auckland,
Auckland, New Zealand
7.09 Pyrans and their Benzo Derivatives: Applications 701
B W FRAVEL, Butler University, Indianapolis, IN, USA
7.10 Thiopyrans and their Benzo Derivatives 72?
J D HEPWORTH, University of Central Lancashire, Preston, UK
B M HERON, University of Leeds, Leeds, UK
7.11 Six-membered Rings with One Selenium or Tellurium Atom 955
F S GUZIEC, Jr. and L J GUZIEC, Southwestern University, Georgetown, TX, USA
7.12 Six-membered Rings with One Phosphorus Atom 1003
G L EDWARDS, The University of New South Wales, Sydney, NSW, Australia
M BALASUBRAMANIAN, Pfizer Inc., Groton, CT, USA
R MURUGAN, Vertellus Specialties Inc., Indianapolis, IN, USA
7.13 Six-membered Rings with One Arsenic, Antimony, or Bismuth Atom 1039
A J ASHE, III, University of Michigan, Ann Arbor, MI, USA
7.14 Six-membered Rings with One Other Element 1049
P NORRIS, Youngstown State University, Youngstown, OH, USA
Index 1067
VOLUME 8 SIX-MEMBERED RINGS WITH TWO HETEROATOMS, AND THEIR
FUSED GARBOCYGLIC DERIVATIVES
8.01 Pyridazines and their Benzo Derivatives 1
B U W MAES and G L F LEMIERE, University of Antwerp, Antwerp, Belgium
8.02 Pyrimidines and their Benzo Derivatives 117
G W REWCASTLE, The University of Auckland, Auckland, New Zealand
8.03 Pyrazines and their Benzo Derivatives 273
N SATO, Yokohama City University, Yokohama, Japan
8.04 1,2-Oxazines and their Benzo Derivatives 3^3
M BALASUBRAMANIAN, Pfizer Inc., Groton, CT, USA
8.05 1,3-Oxazines and their Benzo Derivatives 373
L LAZAR and F FULOP, University of Szeged, Szeged, Hungary
8.06 1,4-Oxazines and their Benzo Derivatives 461
R A AITKEN and K M AITKEN, University of St. Andrews, St. Andrews, UK
8.07 1,2- Fhiazines and their Benzo Derivatives 513
S M WEINREB, Pennsylvania State University, University Park, PA, USA
R K ORR, Schering-Plough Research Institute, Union, NJ, USA
8.08 1,3-Thiazines and their Benzo Derivatives 557
N KARODIA, University of Bradford, Bradford, UK
8.09 1,4-Thiazines and their Benzo Derivatives 607
R A AITKEN and K M AITKEN, University of St. Andrews, St. Andrews, UK
8.10 1,2-Dioxins, Oxathiins, Dithiins, and their Benzo Derivatives 677
E KLEINPETER, Universitdt Potsdam, Potsdam, Germany
Contents xiii
8.11 1,3-Dioxins, Oxathiins, Dithiins, and their Benzo Derivatives 739
E KLEINPETER and M SEFKOW, Umversitat Potsdam, Potsdam, Germany
8.12 1,4-Dioxins, Oxathiins, Dithiins, and their Benzo Derivatives 857
G GUILLAUMET and F SUZENET, Unwersite a Orleans, Orleans, France
Index 907
VOLUME 9 SIX-MEMBERED RINGS WITH THREE OR MORE
HETEROATOMS, AND THEIR FUSED CARBOCYCLIC DERIVATIVES
9.01 1,2,3-Triazines and their Benzo Derivatives 1
D DOPP and H DOPP, Universitiit Duisburg-Essen, Essen, Germany
9.02 1,2,4-Triazines and their Benzo Derivatives 95
V CHARUSHIN, V RUSINOV, and O CHUPAKHIN, Russian Academy of Sciences,
Ekaterinburg, Russia
9.03 1,3,5-Triazines 197
G GIACOMELLI and A PORCHEDDU, University of Sassan, Sassart, Italy
9.04 1,2,3-Oxadiazines and 1,2,3-Thiadiazines 291
M O HUNSEN, Kenyon College, Gambier, OH, USA
9.05 1,2,4-Oxadiazines and 1,2,4-Thiadiazines 301
P NORRIS, Youngstown State University, Youngston, OH, USA
9.06 1,2,5-Oxadiazines and 1,2,5-Thiadiazines 345
G W MORROW, University of Dayton, Dayton, OH, USA
9.07 1,2,6-Oxadiazines and 1,2,6-Thiadiazines 355
P M WEINTRAUB, Warren, NJ, USA
9.08 1,3,4-Oxadiazines and 1,3,4-Thiadiazines 401
W-D PFEIFFER, University of Greifswald, Greifswald, Germany
9.09 1,3,5-Oxadiazines and 1,3,5-Thiadiazines 457
N SHOBANA and P FARID, Abbott Laboratories, Abbott Park, 1L, USA
9.10 Dioxazines, Oxathiazines, and Dithiazines 523
E JUARISTI, B R DIAZ, and J L OLIVARES-ROMERO, Centro de Investigation
y de Estudios Avanzados del Instituto Politecnico National, Mexico City, Mexico
9.11 Six-membered Rings with 1,2,4-Oxygen or Sulfur Atoms 569
E KLEINPETER, Universitiit Potsdam, Potsdam, Germany
9.12 1,2,4,5-Tetrazines 641
B STANOVNIK, U GROSELJ, and J SVETE, University of Ljubljana, Ljubljana,
Slovenia
9.13 Other Tetrazines and Pentazines 715
V BENIN, University of Dayton, Dayton, OH, USA
9.14 Other Six-membered Rings with Four or Five Nitrogen, Oxygen, or Sulfur 737
G L FRANCIS, CSIRO, Melbourne, VIC, Australia
9.15 Six-membered Rings with Two or More Heteroatoms with at least One Selenium
or Tellurium 791
F S GUZIEC, Jr. and L J GUZIEC, Southwestern University, Georgetown, TX, USA
9.16 Six-membered Rings with Two or More Heteroatoms with at least One Phosphorus 835
K AFARINKIA, University of Bradford, Bradford, UK
9.17 Six-membered Rings with Two or More Heteroatoms with at least One Arsenic
to Bismuth 875
A GUVEN, Anadolu University, EskiseAir, Turkey
xjv Contents
9.18 Six-mcmbercd Rings with Two or More Heteroatoms with at least One Silicon to Lead 913
I D LICKISS, Imperial College London, London, UK
9 19 Six-membcred Rings with Two or More Heteroatoms with at least One Boron 961
V D ROMANKNKO, Institute of Bioorganic Chemistry and Petrochemistry, Kiev, Ukraine
J-M SOTIROPOULOS, Universitede Pau et Pays de I Adour, Pau, France
, . 1009
Index
VOLUME 10 RING SYSTEMS WITH AT LEAST TWO FUSED HETEROGYCLIC
FIVE- OR SIX-MEMBERED RINGS WITH NO BRIDGEHEAD HETEROATOM
10.01 Bicyclic 5-5 Systems: Two Heteroatoms 1:1 1
A KRUTOSIKOVA, University of St. Cyril and Methodius, Trnava, Slovakia
T GRACZA, Slovak University of Technology, Bratislava, Slovakia
10.02 Bicyclic 5-5 Systems: Three Heteroatoms 1:2 65
A J MOORE, University of Sunderland, Sunderland, UK
10.03 Bicyclic 5-5 Systems: Four Heteroatoms 1:3 129
Y A JACKSON and N O TOWNSEND, University of West Indies, Jamaica, West Indies
10.04 Bicyclic 5-5 Systems: Four Heteroatoms 2:2 161
J D WILDEN, University College London, London, UK
10.05 Bicyclic 5-5 Systems: Five Heteroatoms 2:3 and Six Heteroatoms 3:3 189
F HEANEY and L DOYLE, National University of Ireland, Maynooth,
Republic of Ireland
10.06 Bicyclic 5-6 Systems: Two Heteroatoms 1:1 263
A R SHERMAN, College of Notre Dame of Maryland, Baltimore, MD, USA
10.07 Bicyclic 5-6 Systems: Three Heteroatoms 1:2 339
T J DELIA, Central Michigan University, Mt. Pleasant, MI, USA
10.08 Bicyclic 5-6 Systems: Three Heteroatoms 2:1 431
B R BUCKLEY, Loughborough University, Loughborough, UK
10.09 Bicyclic 5-6 Systems: Four Heteroatoms 1:3 493
M C ELLIOTT, Cardiff University, Cardiff, UK
10.10 Bicyclic 5-6 Systems: Four Heteroatoms 3:1 511
B R BUCKLEY and S P NEARY, Loughborough University, Loughborough, UK
10.11 Bicyclic 5-6 Systems: Purines 525
I COLLINS and J J CALDVVELL, The Institute of Cancer Research, Sutton, UK
10.12 Bicyclic 5-6 Systems: Other Four Heteroatoms 2:2 599
M H ELNAGDI, Cairo University, Giza, Egypt
N AL-AWADI, University of Kuwait, Safat, Kuwait
I A ABDELHAMID, Cairo University, Giza, Egypt
10.13 Bicyclic 5-6 Systems: Five Heteroatoms 2:3 or 3:2 661
F ALDABBAGH, National University of Ireland, Galway, Republic of Ireland
10.14 Bicyclic 5-6 Systems: Six and Seven Heteroatoms 703
C A RAMSDEN, Keek University, Keek, UK
10.15 Bicyclic 6-6 Systems: Two Heteroatoms 1:1 713
A P DOBBS, Queen Mary, University of London, London, UK
10.16 Bicyclic 6-6 Systems: Three Heteroatoms 1-2 -jzq
E S H EL ASHRY and N RASHED, Alexandria University, Alexandria, Egypt
Contents xv
10.17 Bicyclic 6-6 Systems: Four Heteroatoms 1:3 847
P W GROUNDWATER and R J ANDERSON, University of Sunderland,
Sunderland, UK
M NYERGES, Technical University of Budapest, Budapest, Hungary
10.18 Bicyclic 6-6 Systems: Pteridines 915
C SUCKLING, G GIBSON, and J HUGGAN, University of Strathclyde, Glasgow, UK
10.19 Bicyclic 6-6 Systems: Other Four Heteroatoms 2:2 977
J M HERBERT, Sanofi-Aventis, Alnwtck, UK
10.20 Bicyclic 6-6 Systems: Five or More Heteroatoms 1093
K HEMMING, University of Huddersfield, Huddersfield, UK
10.21 Tricyclic Systems: Central Carbocyclic Ring with Fused Five-membered Rings 1135
A GRAHAM and M ROBINSON, University of Wales Swansea, Swansea, UK
10.22 Tricyclic Systems: Central Carbocyclic Ring with Fused Five- and
Six-membered Rings 1201
M P GROZIAK, California State University, East Bay, Hayward, CA, USA
10.23 Tricyclic Systems: Central Carbocyclic Ring with Fused Six-membered Rings 1229
B R BUCKLEY, Loughborough University, Loughborough, UK
Index 1269
VOLUME 11 BICYCLIC 5-5 AND 5-6 FUSED RING SYSTEMS WITH
AT LEAST ONE BRIDGEHEAD (RING JUNCTION) N
11.01 Bicyclic 5-5 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: No
Extra Heteroatom 1
H DHIMANE, UniversitePans Descartes, Pans, France
G LHOMMET, Universite Pierre et Marie Curie-Paris VI, Paris, France
11.02 Bicyclic 5-5 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: One
Extra Heteroatom 1:0 41
J SUFFERT, Universite Louis Pasteur de Strasbourg, Strasbourg, France
11.03 Bicyclic 5-5 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Two
Extra Heteroatoms 2:0 107
L MICOUIN, CNRS, Pans, France
11.04 Bicyclic 5-5 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Two
Extra Heteroatoms 1:1 133
C OLLIVIER, Universite Paul Cezanne-CNRS, Marseille, France
11.05 Bicyclic 5-5 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Three
Extra Heteroatoms 2:1 199
J MARCO-CONTELLES, Instituto de Quimica Orgdnica General (CSIC), Madrid, Spain
E PEREZ-MAYORAL and P BALLESTEROS, UNED, Madrid, Spain
11.06 Bicyclic 5-5 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Three
Extra Heteroatoms 3:0 307
S SABA and J A CIACCIO, Fordham University, Bronx, NY, USA
11.07 Bicyclic 5-5 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Four
Extra Heteroatoms 2:2 325
J ZHU and L NEUVILLE, Institut de Chimie des Substances Naturelles, CNRS,
Gif-sur-Yvette, France
11.08 Bicyclic 5-5 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Four Extra
Heteroatoms 3:1 351
G HILT, W HESS, and C HENGST, Philipps-Universitat Marburg, Marburg, Germany
xvj Contents
11.09 Bicyclic 5-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: No Extra ^
Heteroatom 0:0 .
A BRANDI and S CICCHI, Universita di Firenze, Sesto Fwrentino, bl, Italy
11.10 Bicyclic 5-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: One Extra
Heteroatom 1:0
F COUTY and G EVANO, Universite de Versailles Satnt-Quentm-en-Yvelines, Versailles,
France
11.11 Bicyclic 5-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: One
Extra Heteroatom 0:1 ¦()
M TADDEI, Universita degli Studi di Siena, Siena, Italy
11.12 Bicyciic 5-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Two
Extra Heteroatoms 1:1 ¦ ¦
A C REGAN, University of Manchester, Manchester, UK
11.13 Bicyclic 5-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Two
Extra Heteroatoms 2:0 589
L BISGHOFF, Equipe de Chimie Organique Fine et Heterocyclique (ECOFH), Rouen,
France
11.14 Bicyclic 5-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Two
Extra Heteroatoms 0:2 629
J RODRIGUEZ and T CONSTANTIEUX, Universite Paul Cezanne (Mx-Marseille III),
Marseille, France
11.15 Bicyclic 5-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Three
Extra Heteroatoms 3:0 645
G HAJOS and Z RIEDL, Institute of Biomokcular Chemistry, Chemical Research Center,
Pusztaszeri ut, Hungary
11.16 Bicyclic 5-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Three
Extra Heteroatoms 2:1 671
G HAJOS and Z RIEDL, Institute of Biomokcular Chemistry, Chemical Research Centre,
Budapest, Hungary
11.17 Bicyclic 5-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Three
Extra Heteroatoms 1:2
G HAJOS and Z RIEDL, Institute of Biomokcular Chemistry, Chemical Research Centre,
Budapest, Hungary
11.18 Bicyclic 5-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Four
Extra Heteroatoms 3:1 #19
G HAJOS and Z RIEDL, Institute of Biomokcular Chemistry, Chemical Research Centre,
Budapest, Hungary
11.19 Bicyclic 5-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Four
Extra Heteroatoms 2:2 §47
G HAJOS and Z RIEDL, Institute of Biomokcular Chemistry, Chemical Research Centre
Budapest, Hungary
11.20 Bicyclic 5-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Four
Extra Heteroatoms 1:3 ^y^
G HAJOS and Z RIE DL, Institute of Biomokcular Chemistry, Chemical Research Centre
Budapest, Hungary
11.21 Bicyclic 5-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom- Five
Extra Heteroatoms 3:2 909
G HAJOS and Z RIEDL, Institute of Biomokcular Chemistry, Chemical Research Centre
Budapest, Hungary
Index
919
Contents xvii
VOLUME 12 FIVE- AND SIX-MEMBERED FUSED SYSTEMS WITH
BRIDGEHEAD (RING JUNCTION) HETEROATOMS CONCLUDED: 6-6
BICYCLIC WITH ONE OR TWO N OR OTHER HETEROATOMS;
POLYCYCLIC; SPIROCYCLIC
12.01 Bicyclic 6-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: No Extra
Heteroatom 1
C AVENDANO and J C MENENDEZ, Universidad Complutense, Madrid, Spain
12.02 Bicyclic 6-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: One
Extra Heteroatom 1:0 77
I HERMECZ and L VASVARI-DEBRECZY, Chinoin Pharmaceutical and Chemical
Works Ltd., Budapest, Hungary
12.03 Bicyclic 6-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Two
Extra Heteroatoms 2:0 219
P MATYUS and P TAPOLCSANYI, Semmelweis University, Budapest, Hungary
12.04 Bicyclic 6-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Two
Extra Heteroatoms 1:1 257
I HERMECZ and L VASVARI-DEBRECZY, Chinoin Pharmaceutical and Chemical
Works Ltd., Budapest, Hungary
12.05 Bicyclic 6-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Three
Extra Heteroatoms 3:0 321
M P MAHAJAN and C MOHAN, Guru Nanak Dev University, Amritsar, India
12.06 Bicyclic 6-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Three
Extra Heteroatoms 2:1 327
M P MAHAJAN, G BHARGAVA, and C MOHAN, Guru Nanak Dev University,
Amritsar, India
12.07 Bicyclic 6-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Four
Extra Heteroatoms 3:1 341
M P MAHAJAN and C MOHAN, Guru Nanak Dev University, Amritsar, India
12.08 Bicyclic 6-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Four
Extra Heteroatoms 2:2 347
M P MAHAJAN, A MARWAHA, and C MOHAN, Guru Nanak Dev University,
Amritsar, India
12.09 Bicyclic 6-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Five
Extra Heteroatoms 3:2 357
M P MAHAJAN and C MOHAN, Guru Nanak Dev University, Amritsar, India
12.10 Bicyclic Systems with Two Bridgehead (Ring Junction) Nitrogen Atoms 365
S RADL, Zentiva - Research Institute for Pharmacy and Biochemistry, Prague,
Czech Republic
12.11 Bicyclic Systems with Bridgehead (Ring Junction) Sulfur, Selenium,
or Tellurium Atoms 481
I FORRISTAL, King Fahd University of Petroleum Minerals, Dhahran, Saudi Arabia
12.12 Bicyclic Systems with Bridgehead (Ring Junction) Phosphorus, Arsenic,
Antimony, or Bismuth Atoms 527
S SCHWIKKARD, Kingston University, Kingston, UK
12.13 Bicyclic Systems with Bridgehead (Ring Junction) Boron Atoms 573
Yu N BUBNOV, M E GURSKII, and S Yu ERDYAKOV, Russian Academy of
Sciences, Moscow, Russia
12.14 Three Heterocyclic Rings Fused (5-5-5) 635
K C MAJUMDAR and S K CHATTOPADHYAY, University of Kalyani, Kalyani, India
xviii Contents
12.15 Three Heterocyclic Rings Fused (5-6-5)
S HILTON, The Institute of Cancer Research, Sutton, UK
S ROSSITER, University of Hertfordshire, Hatfield, UK
12.16 Three Heterocyclic Rings Fused (5-5-6)
R L RIGGS, BASF AG, Ludwigshafen, Germany
D M SMITH, University of St Andrews, St Andrews, UK
12.17 Three Heterocyclic Rings Fused (5-6-6) 857
R L RIGGS, BASF AG, Ludwigshafen, Germany
D M SMITH, University of St. Andrews, St. Andrews, UK
12.18 Three Heterocyclic Rings Fused (6-5-6) 975
L STRFKOWSKI, J SACZEWSKI, and M HENARY, Georgia State University,
Atlanta, GA, USA
12.19 Three Heterocyclic Rings Fused (6-6-6) 1007
L STREKOWSKI, M HENARY, and M MOJZYCH, Georgia State University,
Atlanta, GA, USA
12.20 Systems with a Spirocyclic Heteroatom 1037
N M AHMAD, The Institute of Cancer Research, Sutton, UK
Z.Z Compounds containing a Spiro Phosphorus Atom 1065
N A WILLIAMS, Kingston University, Kingston upon Thames, UK
Index 1127
VOLUME 13 SEVEN-MEMBERED HETEROCYCLIC RINGS AND THEIR FUSED
DERIVATIVES
13.01 Azepines and their Fused-ring Derivatives 1
J B BREMNER, University of Wollongong, Wollongong, NSW, Australia
S SAMOSORN, Srinakharinwirot University, Bangkok, Thailand
13.02 Oxepanes and Oxepines 45
L I BELEN KII, Russian Academy of Sciences, Moscow, Russia
13.03 Thiepanes and Thiepines 97
S YAMAZAKI, Nara University of Education, Nara, Japan
13.04 1,2-Diazepines 143
T P MEAGHER, TEKA Consulting, Indianapolis, IN, USA
R MURUGAN, Vertellus Specialties Inc, Indianapolis, IN, USA
13.05 1,3-Diazepines j^j
W M DE BORGGRAEVE and A M VAN DEN BOGAERT, K ULeuven,
I*liven, Belgium
13.06 1,4-Diazepines jg-^
N A MEANWELL and M A WALKER, Bristol-Myers Squibb Research and
Development, Wallingford, CT, USA
13.07 1,2-Oxazepines and 1,2-Thiazepines ?37
J B BREMNER, University of Wollongong, Wollongong, NSW, Australia
S SAMOSORN, Srinakharinwirot University, Bangkok, Thailand
13.08 1,3-Oxazepines and 1,3-Thiazepines 245
Jc *ISScI^ER University °f Wollongong, Wollongong, NSW, Australia
b SAMOSORN, Snnakhartnwirot University, Bangkok, Thailand
13.09 1,4-Oxazepines and 1,4-Thiazepines 2SS
W DEHAEN and T H NGO, University of Leuven, Leuven, Belgium
Contents xix
13.10 1,2-Dioxepanes, 1,2-Oxathiepanes, and 1,2-Dithiepanes 299
M J HADDADIN and C J NACHEF, American University of Beirut, Beirut,
Lebanon
13.11 1,3-Dioxepanes, 1,3-Oxathiepanes, and 1,3-Dithiepanes 321
H FRAUENRATH and S FLOCK, University of Kassel, Kassel, Germany
13.12 1,4-Dioxepanes, 1,4-Oxathiepanes, and 1,4-Dithiepanes 367
H FRAUENRATH and S FLOCK, Universitat GH Kassel, Kassel, Germany
R MURUGAN, Vertellus Specialties Inc., Indianapolis, IN, USA
E F V SCRIVEN, University of Florida, Gainesville, FL, USA
13.13 Seven-membered Rings with Three Heteroatoms 1,2,3 387
A KISELYOV and A KHVAT, ChemDw Inc., San Diego, CA, USA
13.14 Seven-membered Rings with Three Heteroatoms 1,2,4 399
G I YRANZO and E L MOYANO, Universidad Nacwnal de Cordoba, Cordoba,
Argentina
13.15 Seven-membered Rings with Three Heteroatoms 1,2,5 433
R RANJITH KUMAR and S PERUMAL, Madurai Kamaraj University,
Madurai, India
M BALASUBRAMANIAN, Pfizer, Inc., Groton, CT, USA
13.16 Seven-membered Rings with Three Heteroatoms 1,3,5 489
0 V DENISKO, Chemical Abstracts Service, Columbus, OH, USA
13.17 Seven-membered Rings with Four or More Heteroatoms 529
G N NIKONOV, Alchem Laboratories Co., Alachua, FL, USA
Index 571
VOLUME 14 EIGHT-MEMBERED AND LARGER HETEROCYGLIC RINGS
AND THEIR FUSED DERIVATIVES, OTHER SEVEN-MEMBERED RINGS
14.01 Eight-membered Rings with One Nitrogen Atom 1
D C ONICIU, University of Florida, Gainesville, FL, USA
14.02 Eight-membered Rings with One Oxygen Atom 49
A M S SILVA and A C TOME, University of Aveiro, Aveiro, Portugal
14.03 Eight-membered Rings with One Sulfur Atom 89
H ECKERT, Technical University of Munich, Garching, Germany
14.04 Eight-membered Rings with Two Heteroatoms 1,2 99
G CIRRINCIONE and P DIANA, Universitd degli Studi di Palermo, Palermo, Italy
14.05 Eight-membered Rings with Two Heteroatoms 1,3 169
G CIRRINCIONE and P DIANA, Universitd degli Studi di Palermo, Palermo, Italy
14.06 Eight-membered Rings with Two Heteroatoms 1,4 255
1 SHCHERBAKOVA, MediProPharma, Inc., Midvale, (IT, USA
14.07 Eight-membered Rings with Two Heteroatoms 1,5 303
G CIRRINCIONE and P DIANA, Universitd degli Studi di Palermo, Palermo, Italy
14.08 Eight-membered Rings with Three Heteroatoms 475
D O TYMOSHENKO, Albany Molecular Research, Inc., Albany, NY, USA
14.09 Eight-membered Rings with Four or More Heteroatoms 517
I SHCHERBAKOVA, MediProPharma, Inc., Midvale, UT, USA
14.10 Nine-membered Rings 547
D O TYMOSHENKO, AMRI, Albany, NY, USA
xx Contents
14.11 Ten-membered Rings or Larger with One or More Nitrogen Atoms 613
P HERMANN and J KOTEK, Universita Karlova, Prague, Czech Republic
14.12 Ten-membered Rings or Larger with One or More Oxygen Atoms 667
S PAPPALARDO, Universita di Catania, Catania, Italy
M F PARISI, Universita di Messina, Messina, Italy
14.13 Ten-membered Rings or Larger with One or More Sulfur Atoms 751
H ECKERT, Technical University of Munich, Garching, Germany
M ROLLER, Bundeswehr Institute of Pharmacology and Toxicology, Munich, Germany
14.14 Ten-membered Rings or Larger with One or More Nitrogen and Oxygen
and/or Sulfur Atoms 803
G W GOKEL and E K ELLIOTT, Washington University School of Medicine,
St. Louis, MO, USA
14.15 Ten-membered Rings or Larger with One or More Oxygen and Sulfur Atoms 829
Y HABATA, Toho University, Chiba, Japan
14.16 Rings containing Selenium or Tellurium 863
G L SOMMEN, Lonza AG, Walliser Werke, Visp, Switzerland
14.17 Rings containing Phosphorus 901
A M SHESTOPALOV, Zelinsky Institute of Organic Chemistry, Moscow, Russia
A A SHESTOPALOV, Duke University, Durham, NC, USA
14.18 Rings containing Arsenic, Antimony, or Bismuth 945
V D ROMANENKO, Institute of Bioorganic Chemistry and Petrochemistry, Kiev, Ukraine
J-M SOTIROPOULOS, Universite de Pau et Pays de I Adour, Pau, France
14.19 Rings containing Silicon to Lead 979
F SACZEWSKI and A KORNICKA, Medical University of Gdansk, Gdansk, Poland
14.20 Rings containing Boron 10}9
G V MORROW, University of Dayton, Dayton, OH, USA
14.21 Rings containing Other Elements 1051
T P MEAGHER, TEKA Consulting, Indianapolis, IN, USA
14.22 Multiple Macroheterocyclic Rings 1071
A M-P PEDERSON and H W GIBSON, Virginia Polytechnic Institute and State
University, Blacksburg, VA, USA
Indt X 1087
VOLUME 15 CUMULATIVE SUBJECT INDEX !
.«*
«?
Introduction
Alan R. Katritzky, Christopher A. Ramsden, Eric F. V. Scriven, and Richard J. K. Taylor
1 Scope, Significance, and Aims 50
1.1 Scope 50
1.2 Significance 50
1.3 Aims of CHEC-I, CHEC-II and CHEC-III 50
2 Arrangement of the Work in Volumes 51
2.1 Relationship of CHEC-III to CHEC-I and CHEC-II 51
2.2 Arrangement of CHEC-III in Volumes 51
2.3 Arrangement of CHEC-II in Volumes 51
2.4 Arrangement of CHEC-I in Volumes 52
3 Rationale for Arrangement of Material in Individual Volumes 52
3.1 Major Divisions of Carbocyclic and Heterocyclic Chemistry 52
3.2 Saturated Heterocyclic Compounds 53
3.3 Partially Unsaturated Heterocyclic Compounds 53
3.4 Heteroaromatic Compounds 53
3.5 Characteristics of Heteroatoms in Rings 53
3.6 The General Chapters of CHEC-I 54
4 Organization of Individual Monograph Chapters 54
4.1 Introduction 55
4.2 Theoretical Methods 55
4.3 Experimental Structural Methods 55
4.4 Thermodynamic Aspects 55
4.5 Reactivity of Fully Conjugated Rings 55
4.6 Reactivity of Nonconjugated Rings 56
4.7 Reactivity of Substituents Attached to Ring Carbon Atoms 56
4.8 Reactivity of Substituents Attached to Ring Heteroatoms 56
4.9 Ring Syntheses Classified by Number of Ring Atoms in Each Component 56
4.10 Ring Synthesis by Transformation of Another Ring 56
4.11 Synthesis of Particular Classes of Compounds and Critical Comparison of the Various
Routes Available 56
4.12 Important Compounds and Applications 56
5 The Reference System 56
6 The Indexes 57
6.1 Ring Index 57
6.2 Subject Index 57
|
adam_txt |
Contents of All Volumes
VOLUME 1 THREE-MEMBERED HETEROCYCLES, TOGETHER WITH
ALL FUSED SYSTEMS CONTAINING A THREE-MEMBERED
HETEROCYCLIG RING
1.01 Aziridines and Azirines: Monocyclic 1
A PADWA, Emory University, Atlanta, GA, USA
1.02 Aziridines and Azirines: Fused-ring Derivatives 105
M C McMILLS and S C BERGMEIER, Ohio University, Athens, OH, USA
1.03 Oxiranes and Oxirenes: Monocyclic 173
G DAKE, University of British Columbia, Vancouver, BC, Canada
1.04 Oxiranes and Oxirenes: Fused-ring Derivatives 235
D M HODGSON, University of Oxford, Oxford, UK
M A H STENT, Key Orgamcs Ltd., Cornwall, UK
1.05 Thiiranes and Thiirenes: Monocyclic 299
J WARKENTIN, McMaster University, Hamilton, ON, Canada
D PLAZUK, University of Lodz, Lodz, Poland
1.06 Thiiranes and Thiirenes: Fused-ring Derivatives 391
T VILAIVAN, W CHAVASIRI, and P RASHATASAKHON, Chulalongkorn University,
Bangkok, Thailand
1.07 Three-membered Rings with One Selenium or Tellurium Atom 433
R S GLASS, The University of Arizona, Tucson, AZ, USA
1.08 Phosphiranes, Phosphirenes, and Heavier Analogues 457
H HEYDT, Technische Universitdt Kaiserslautern, Kaiserslautern, Germany
1.09 Three-membered Rings with One Silicon, Germanium, Tin or Lead Atom 483
M A MENDEZ-ROJAS, Universidadde las Americas, Cholula, Mexico
G MERINO, Universidad de Guanajuato, Guanajuato, Mexico
1.10 Three-membered Rings with One Boron Atom 513
N FARFAN, Universidad'National Autonoma de Mexico, Mexico City, Mexico
H I BELTRAN, Universidad Autonoma Metropolitana, Cuajimalpa, Mexico City, Mexico
1.11 Diaziridines and Diazirines 539
G D McALLISTER, A PERRY, and R J K TAYLOR, University of York, York, UK
1.12 Oxaziridines and Oxazirines 559
F A DAVIS, Temple University, Philadelphia, PA, USA
B-C CHEN, Bristol-Myers Squib/? Company, Princeton, NJ, USA
P ZHOU, Wyeth Research, Princeton, NJ, USA
v
vj Contents
1.13 Thiaziridines and Thiazirenes
U ZOLLRR, Haifa University - Oranim, Kiryat Tivon, Israel
1 14 Three-membered Rings with Two Oxygen and/or Sulfur Atoms 641
M ROJE and T PORTADA, Ructer Boskovic Institute, Zagreb, Croatia
1.15 Three-membered Rings with Two Heteroatoms including Selenium or Tellurium;
Three-membered Rings with Three Heteroatoms °79
L NYULASZI and Z BENKO, Budapest University of Technology
and Economics, Budapest, Hungary
1.16 Three-membered Rings with Two Heteroatoms including Phosphorus to Bismuth 695
L WEBER, Unhersitat Bielefeld, Bielefeld, Germany
1.17 Three-membered Rings with Two Heteroatoms including Other Elements 749
T M GILBERT, Northern Illinois University, DeKalb, IL, USA
Index 79-S
VOLUME 2 FOUR-MEMBERED HETEROCYCLES TOGETHER WITH
ALL FUSED SYSTEMS CONTAINING A FOUR-MEMBERED
HETEROCYCLIC RING
2.01 Azetidines, Azetines and Azetes: Monocyclic 1
G S SINGH, University of Botswana, Gaborone, Botswana
M D'HOOGHE, Ghent University, Ghent, Belgium
N DE KIMPE, Ghent University, Ghent, Belgium
2.02 Cephalosporins 111
B ALCAIDE and C ARAGONCILLO, Unwersidad Complutense de Madrid, Madrid, Spain
P ALMENDROS, Instituto de Quimica Orgdnica General, CSIC, Madrid, Spain
2.03 Penicillins 173
J MARCHAND-BRYNAERTand C BRULE, Umversite catholtque de Louvain,
l.ouvain-la-Neuve, Belgium
2.04 Other Fused Azetidines, Azetines and Azetes 239
L K MEHTA and J PARRICK, Brunei University, Uxbridge, UK
2.05 Oxetanes and Oxetenes: Monocyclic 321
H C HAILES, University College London, London, UK
J M BEHRENDT, Aston University, Birmingham, UK
2.06 Oxetanes and Oxetenes: Fused-ring Derivatives 365
P H DUSSAULT and C XU, University of Nebraska - Lincoln, Lincoln, NE, USA
2.07 Thietanes and Thietes: Monocyclic 389
S LESNIAK, W J KINART, and J LEWKOWSKI, University of Lodz, Lodz, Poland
2.08 Thietanes and Thietes: Fused-ring Derivatives 429
S LESNIAK, W J KINART, and J LEWKOWSKI, University of Lodz, Lodz, Poland
2.09 Four-membered Rings with One Selenium or Tellurium Atom 463
M KOKKTSU and H ISHIHARA, Gifu University, Gifu, Japan
2.10 Four-membered Rings with One Phosphorus, Arsenic, Antimony, or Bismuth Atom 479
I KAWASHIMA and J KOBAYASHI, The University of Tokyo, Tokyo, Japan
2.11 Four-membered Rings with One Silicon, Germanium, Tin, or Lead Atom 511
M V KOZYTSKA and G B DUDLEY, The Florida State University, Tallahasee, FL, USA
ZM Four-membered Rings with One Boron or Other Atom c55
\1 \IORITA, R C BAUER, and j M STRYKER, University of Alberta, Edmonton
AB, Canada
i
I
Contents vii
2.13 Four-membered Rings with Two Nitrogen Atoms 623
B B LOHRAY and V B LOHRAY, Bhuvid Research Laboratory, Pvt. Ltd.,
Ahmedabad, India
B K SRIVASTAVA, Zydus Research Center, Ahmedabad, India
2.14 Four-membered Rings with One Oxygen and One Nitrogen Atom 689
S FLORIO, V CAPRIATI, and R LUISI, Universitd di Ban, Ban, Italy
2.15 Four-membered Rings with One Sulfur and One Nitrogen Atom 713
P HUDHOMME, UniversitedAngers, Angers, France
2.16 Four-membered Rings with Two Oxygen Atoms 775
D K TAYLOR, The University of Adelaide, Adelaide, SA, Australia
2.17 Four-membered Rings with One Oxygen and One Sulfur Atom 795
D K TAYLOR, The University of Adelaide, Adelaide, SA, Australia
2.18 Four-membered Rings with Two Sulfur Atoms 811
J DRABOWIQZ, Polish Academy of Sciences, Czestochowa, Poland, Jan Dlugosz University
of Czestochowa, Czestochowa, Poland
J LEWKOWSKI, University of Lodz, Lodz, Poland
W KUDELSKA, Jan Dlugosz University of Czestochowa, Czestochowa, Poland
A ZAJAC, Polish Academy of Sciences, Lodz, Poland
2.19 Four-membered Rings with Two or More Heteroatoms including Selenium
or Tellurium 853
T SHIMIZU, Tokyo Metropolitan University, Tokyo, Japan
2.20 Four-membered Rings with Two Heteroatoms including Phosphorus to Bismuth 875
U ZENNECK and M HOFMANN, University of Erlangen-Nurnberg, Erlangen, Germany
2.21 Four-membered Rings with Two Heteroatoms including Silicon to Lead 907
M CYPRYK, Polish Academy of Sciences, Lodz, Poland
A JOZWIAK, University of Lodz, Lodz, Poland
2.22 Four-membered Rings with Three Heteroatoms with at least One Oxygen,
Sulfur or Nitrogen Atom 939
A SACKUS, Kaunas University of Technology, Kaunas, Lithuania
F A SL0K, Vipergen ApS, Copenhagen, Denmark
2.23 Four-membered Rings with Three Heteroatoms not including Oxygen,
Sulfur or Nitrogen Atom 973
E LUKEVICS and E ABELE, Latvian Institute of Organic Synthesis, Riga, Latvia
Index 991
VOLUME 3 FIVE-MEMBERED RINGS WITH ONE HETEROATOM
TOGETHER WITH THEIR BENZO AND OTHER CARBOCYGLIG-FUSED
DERIVATIVES
3.01 Pyrroles and their Benzo Derivatives: Structure 1
M D'ISCHIA, A NAPOLITANO, and A PEZZELLA, University of Naples
"Federico II", Naples, Italy
3.02 Pyrroles and their Benzo Derivatives: Reactivity 45
B A TROFIMOV and N A NEDOLYA, Russian Academy of Sciences - Siberian
Branch, Irkutsk, Russia
3.03 Pyrroles and their Benzo Derivatives: Synthesis 269
J BERGMAN and T JANOSIK, Karolinska Institute, Huddinge, Sweden
3.04 Pyrroles and their Benzo Derivatives: Applications 353
M D'ISCHIA, A NAPOLITANO and A PEZZELLA, University of Naples "Federico II",
Naples, Italy
vjj! Contents
ion
3.05 Furans and their Benzo Derivatives: Structure Joy
A SKNNING, Technical University of Denmark, Kgs. Lyngby, Denmark
3 06 Furans and their Benzo Derivatives: Reactivity 407
H N C WONG, The Chinese University of Hong Kong, Hong Kong, People's Republic of China
K-S YEUNG, Bristol-Myers Squibb Pharmaceutical Research Institute, Wallingford, CT, USA
Z YANG, Peking University, Beijing, People's Republic of China
3.07 Furans and their Benzo Derivatives: Synthesis 497
T GRAENING and F THRUN, TU Berlin, Berlin, Germany
3.08 Furans and their Benzo Derivatives: Applications 571
B A KEAY and J M HOPKINS, University of Calgary, Calgary, AB, Canada
P W DIBBLE, University of Lethbridge, Lethbridge, AB, Canada
3.09 Thiophenes and their Benzo Derivatives: Structure 625
P MOLINA, A ARQUES, and I CARTAGENA, University of Murcia, Murcia, Spain
3.10 Thiophenes and their Benzo Derivatives: Reactivity 741
S RAJAPPA, B-l, Melody Apartments, ICS Colony, Pune 411007, India
A R DESHMUKH, National Chemical Laboratory, Pune, India
3.11 Thiophenes and their Benzo Derivatives: Synthesis 843
O SATO and J NAKAYAMA, Saitama University, Saitama, Japan
3.12 Thiophenes and their Benzo Derivatives: Applications 931
J SCHATZ, T BRENDGEN, and D SCHUHLE, University of Ulm, Ulm, Germany
3.13 Selenophenes 975
F T PELKEY, Hobart and William Smith Colleges, Geneva, NY, USA
3.14 Tellurophenes 1007
V I MINKIN and I D SADEKOV, Rostov State University, Rostov on Don, Russia
3.15 Phospholes 1029
R REAU, University of Rennes 1, Rennes, France
P W DYER, Durham University, Durham, UK
3.16 Arsoles, Stiboles, and Bismoles U49
V MILATA, Slovak Technical University, Bratislava, Slovakia
3.17 Siloles, Germoles, Stannoles, and Plumboles 1181
B WRACKMEYER and O L TOK, Universitdt Bayreuth, Bayreuth, Germany
3.18 Boroles j 22S
G VARVOUNIS, University of loannina, loannina, Greece
3.19 Five-membered Rings with Other Elements 1243
A P SADIMENKO, University of Fort Hare, Alice, South Africa
lndex 1305
VOLUME 4 FIVE-MEMBERED RINGS WITH TWO HETPROATOMS
EACH WITH THEIR FUSED GARBOCYCLIG DERIVATIVES
4.01 Pyrazoles
L "\ET, Albany Molecular Research, Inc., Albany, NY, USA
4.02 Imida/oles
N XI, Q HUANG, and L LIU, Amgen, Inc., Thousand Oaks, CA, USA
4.03 Isoxazoles
F MArHiaTX,F /MCORDERO' U™ersita di Firenze, Sesto Fiorentmo, Italy ^
r Aim.Ht. i 11, Istituto di chimica dei composti organometallki del CNR Sesto
riorenttno, Italy '
Contents ix
4.04 Oxazoles 487
V YEH, Astellas Research Institute of America, Skokie, IL, USA
R IYENGAR, Enanta Pharmaceuticals Inc., Watertown, MA, USA
4.05 Isothiazoles 545
F CLERICI, M L GELMI, and S PELLEGRINO, Universita di Mi/ano, Milan, Italy
4.06 Thiazoles 635
B CHEN and W HEAL, The University of Sheffield, Sheffield, UK
4.07 1,2-Selenazoles 755
J MLOCHOWSKI, Wroclaw University of Technology, Wroclaw, Poland
4.08 1,3-Selenazoles 791
M KOKETSU and H ISHIHARA, Gifu University, Gifu, Japan
4.09 1,2-Dioxoles and 1,2-Oxathioles 823
R A AITKEN and L A POWER, University of St. Andrews, St. Andrews, UK
4.10 1,3-Dioxoles and 1,3-Oxathioles 841
R A AITKEN and L A POWER, University of St. Andrews, St. Andrews, UK
4.11 1,2-DithioIes 893
R MARKOVIC and A RASOVIC, University of Belgrade, Belgrade, Serbia
4.12 1,3-Dithioles 955
P BALGZEWSKI, Centre of Molecular and Macromolecular Studies PAS Lodz, Poland
W KUDELSKA, Jan Dtugosz University (JDU), Cz§stochowa, Poland
A BODZIOGH, Centre of Molecular and Macromolecular Studies PAS Lodz, Poland
4.13 Five-membered Rings with Two Adjacent Heteroatoms with at least One Selenium
or Tellurium 1091
M B NIELSEN, University of Copenhagen, Copenhagen, Denmark
4.14 Five-membered Rings with Two Nonadjacent Heteroatoms with at least One
Selenium or Tellurium 1119
M B NIELSEN, University of Copenhagen, Copenhagen, Denmark
4.15 Five-membered Rings with Two Adjacent Heteroatoms with at least One
Phosphorus, Arsenic, or Antimony 1155
K KARAGHIOSOFF, Ludwig-Maximilians Universitat, Munich, Germany
4.16 Five-membered Rings with Two Nonadjacent Heteroatoms with at least One
Phosphorus, Arsenic, or Antimony 1169
J A JOULE, The University of Manchester, Manchester, UK
4.17 Five-membered Rings with Two Adjacent Heteroatoms with at least One Boron 1189
A J ASHE, III, University of Michigan, Ann Arbor, MI, USA
4.18 Five-membered Rings with Two Nonadjacent Heteroatoms with at least One Boron 1225
G VARVOUNIS, University of Ioannina, loannina, Greece
4.19 Five-membered Rings with Two Adjacent Heteroatoms with at least One
Other Element 1243
C CANO-SOUMILLAC, Northern Institute for Cancer Research, Newcastle-upon-Tyne, UK
4.20 Five-membered Rings with Two Nonadjacent Heteroatoms with at least One
Other Element 1271
C CANO-SOUMILLAC, Northern Institute for Cancer Research, Newcastle-upon-Tyne, UK
Index 1305
x Contents
VOLUME 5 FIVE-MEMBERED RINGS: TRIAZOLES, OXADIAZOLES
THIADIAZOLES AND THEIR FUSED GAJRBOCYCLIC DERIVATIVES
5.01 1,2,3-Triazoles !
S RACHWAL, Cortex Pharmaceuticals, Inc., Irvine, CA, USA
A R KATRITZKY, University of Florida, Gainesville, FL, USA
5.02 1,2,4-Triazoles K
A D M CURTIS and N JENNINGS, Keele University, Keele, UK
5.03 1,2,3-Oxadiazoles 211
VV FRASER, Aston University, Birmingham, UK
5.04 1,2,4-Oxadiazoles 243
K HEMMING, University of Huddersfield, Huddersfield, UK
5.05 1,2,5-Oxadiazoles 315
G NIKONOV and S BOBROV, Alchem Laboratories Co., Alachua, FL, USA
5.06 1,3,4-Oxadiazoles 397
J SUWINSKI and W SZCZEPANKIEWICZ, Silesian University of Technology,
Gliwice, Poland
5.07 1,2,3-Thiadiazoles 467
D J WILKINS, Key Organics Limited, Camelford, UK
5.08 1,2,4-ThiadiazoIes 487
D J WILKINS, Key Organics Limited Camelford, UK
5.09 1,2,5-Thiadiazoles 515
P A KOUTENTIS, University of Cyprus, Nicosia, Cyprus
5.10 1,3,4-Thiadiazoles 567
P A KOUTENTIS, University of Cyprus, Nicosia, Cyprus
C P CONSTANTINIDES, The University of Cambridge, Cambridge, UK
Index 607
VOLUME 6 OTHER FIVE-MEMBERED RINGS WITH THREE OR MORE
HETEROATOMS, AND THEIR FUSED CARBOCYGLIC DERIVATIVES
6.01 l,2-Oxa/thia-3-azoles 1
O A RAKITIN, Zelinski Institute of Organic Chemistry, Moscow, Russia
6.02 l,3-Oxa/thia-2-azoles 37
C) A RAKITIN, Zelinsky Institute of Organic Chemistry, Moscow, Russia
6.03 l,2-Oxa/thia-4-azoles 6J
N N MAKHOVA, Zelinsky Institute of Organic Chemistry, Moscow, Russia
6.04 l,4-Oxa/thia-2-azoles jq5
N G ARGYROPOULOS, Aristotle University ofThessaloniki, Thessaloniki, Greece
6.05 Fiye-membered Rings with Three Oxygen or Sulfur Atoms in 1,2,3-Positions 145
V \ SAMOSHIN, University of the Pacific, Stockton, CA, USA
6.06 Five-membered Rings with Three Oxygen or Sulfur Atoms in 1,2,4-Positions 191
1 S BALABAN, Karlsruhe Institute of Technology, Karlsruhe, Germany
A 1 BALABAN, Texas A M University at Galveston, Galveston, IX USA
6.07 Tetrazoles
lAf?f ?r ??' V ^OLDOBSKII »d R E TRIFONOV, Si. Petersburg State
Institute of Technology, St. Petersburg, Russia
Contents xi
6.08 Oxatriazoles 425
W FRASER, Aston University, Birmingham, UK
6.09 1,2,3,4-Thiatriazoles 441
W DEHAEN, University of Leuven, Leuven, Belgium
V A BAKULEV, The Urals State Technical University, Ekaterinburg, Russia
6.10 1,2,3,5-Thiatriazoles 485
V A BAKULEV, The Urals State Technical University, Ekaterinburg, Russia
W DEHAEN, University of Leuven, Leuven, Belgium
6.11 1,2,3,5-Dithiadiazoles and 1,3,2,4-Dithiadiazoles 499
R J PEARSON, Keele University, Keele, UK
6.12 Three or Four Heteroatoms including at least One Selenium or Tellurium 517
S YAMAZAKI, Nara University of Education, Nara, Japan
6.13 Three or Four Heteroatoms including at least One Phosphorus 583
V V ZHDANKIN, University of Minnesota Duluth, Duluth, MN, USA
6.14 Three or Four Heteroatoms including at least One Arsenic or Antimony 603
A SCHMIDPETER and K KARAGHIOSOFF, Ludwig-Maximilians-Universitat, Munich,
Germany
6.15 Three or Four Heteroatoms including at least One Boron 615
MVR REDDY, J S CHANDRA, and V J REDDY, University of Minnesota Duluth,
Duluth, MN, USA
6.16 Three or Four Heteroatoms including at least One Silicon 655
T MULLER, Carl von Ossietzky University Oldenburg, Oldenburg, Germany
6.17 Three or Four Heteroatoms including at least One Other Element 691
V N NEMYKIN, University of Minnesota Duluth, Duluth, MN, USA
6.18 Pentazoles 739
T M KLAPOTKE and A HAMMERL, Ludwig-Maximilians Unwersitat Munchen,
Munich, Germany
Index 759
VOLUME 7 SIX-MEMBERED RINGS WITH ONE HETEROATOM, AND THEIR
FUSED GARBOGYCLIC DERIVATIVES
7.01 Pyridines and their Benzo Derivatives: Structure 1
J B HARPER, University of New South Wales, Sydney, NSW, Australia
7.02 Pyridines and their Benzo Derivatives: Reactivity at the Ring 41
D L COMINS, North Carolina State University, Raleigh, NC, USA
S O'CONNOR, Clemson University, Clemson, SC, USA
R S AL-AWAR, Eli Lilly and Company, Indianapolis, IN, USA
7.03 Pyridines and their Benzo Derivatives: Reactivity of Substituents 101
V CAPRIO, University of Auckland, Auckland, New Zealand
7.04 Pyridines and their Benzo Derivatives: Reactivity of Reduced Compounds 171
D BARKER, The University of Auckland, Auckland, New Zealand
7.05 Pyridines and their Benzo Derivatives: Synthesis 217
P A KELLER, University ofWollongong, Wollongong, NSW, Australia
7.06 Pyridines and their Benzo Derivatives: Applications 309
C H MCATEER, Vertellus Specialties Inc., Indianapolis, IN, USA
M BALASUBRAMANIAN, Pfizer Inc., Groton, CT, USA
R MURUGAN, Vertellus Specialties Inc., Indianapolis, IN, USA
xjj Contents
7 07 Pyrans and their Benzo Derivatives: Structure and Reactivity 337
A J PHILLIPS, J A HENDERSON, and K L JACKSON, University of Colorado,
Boulder, CO, USA
7 08 Pyrans and their Benzo Derivatives: Synthesis
M A BRIMBLE, J S GIBSON, and J SPERRY, The University of Auckland,
Auckland, New Zealand
7.09 Pyrans and their Benzo Derivatives: Applications 701
B W FRAVEL, Butler University, Indianapolis, IN, USA
7.10 Thiopyrans and their Benzo Derivatives 72?
J D HEPWORTH, University of Central Lancashire, Preston, UK
B M HERON, University of Leeds, Leeds, UK
7.11 Six-membered Rings with One Selenium or Tellurium Atom 955
F S GUZIEC, Jr. and L J GUZIEC, Southwestern University, Georgetown, TX, USA
7.12 Six-membered Rings with One Phosphorus Atom 1003
G L EDWARDS, The University of New South Wales, Sydney, NSW, Australia
M BALASUBRAMANIAN, Pfizer Inc., Groton, CT, USA
R MURUGAN, Vertellus Specialties Inc., Indianapolis, IN, USA
7.13 Six-membered Rings with One Arsenic, Antimony, or Bismuth Atom 1039
A J ASHE, III, University of Michigan, Ann Arbor, MI, USA
7.14 Six-membered Rings with One Other Element 1049
P NORRIS, Youngstown State University, Youngstown, OH, USA
Index 1067
VOLUME 8 SIX-MEMBERED RINGS WITH TWO HETEROATOMS, AND THEIR
FUSED GARBOCYGLIC DERIVATIVES
8.01 Pyridazines and their Benzo Derivatives 1
B U W MAES and G L F LEMIERE, University of Antwerp, Antwerp, Belgium
8.02 Pyrimidines and their Benzo Derivatives 117
G W REWCASTLE, The University of Auckland, Auckland, New Zealand
8.03 Pyrazines and their Benzo Derivatives 273
N SATO, Yokohama City University, Yokohama, Japan
8.04 1,2-Oxazines and their Benzo Derivatives 3^3
M BALASUBRAMANIAN, Pfizer Inc., Groton, CT, USA
8.05 1,3-Oxazines and their Benzo Derivatives 373
L LAZAR and F FULOP, University of Szeged, Szeged, Hungary
8.06 1,4-Oxazines and their Benzo Derivatives 461
R A AITKEN and K M AITKEN, University of St. Andrews, St. Andrews, UK
8.07 1,2- Fhiazines and their Benzo Derivatives 513
S M WEINREB, Pennsylvania State University, University Park, PA, USA
R K ORR, Schering-Plough Research Institute, Union, NJ, USA
8.08 1,3-Thiazines and their Benzo Derivatives 557
N KARODIA, University of Bradford, Bradford, UK
8.09 1,4-Thiazines and their Benzo Derivatives 607
R A AITKEN and K M AITKEN, University of St. Andrews, St. Andrews, UK
8.10 1,2-Dioxins, Oxathiins, Dithiins, and their Benzo Derivatives 677
E KLEINPETER, Universitdt Potsdam, Potsdam, Germany
Contents xiii
8.11 1,3-Dioxins, Oxathiins, Dithiins, and their Benzo Derivatives 739
E KLEINPETER and M SEFKOW, Umversitat Potsdam, Potsdam, Germany
8.12 1,4-Dioxins, Oxathiins, Dithiins, and their Benzo Derivatives 857
G GUILLAUMET and F SUZENET, Unwersite a"Orleans, Orleans, France
Index 907
VOLUME 9 SIX-MEMBERED RINGS WITH THREE OR MORE
HETEROATOMS, AND THEIR FUSED CARBOCYCLIC DERIVATIVES
9.01 1,2,3-Triazines and their Benzo Derivatives 1
D DOPP and H DOPP, Universitiit Duisburg-Essen, Essen, Germany
9.02 1,2,4-Triazines and their Benzo Derivatives 95
V CHARUSHIN, V RUSINOV, and O CHUPAKHIN, Russian Academy of Sciences,
Ekaterinburg, Russia
9.03 1,3,5-Triazines 197
G GIACOMELLI and A PORCHEDDU, University of Sassan, Sassart, Italy
9.04 1,2,3-Oxadiazines and 1,2,3-Thiadiazines 291
M O HUNSEN, Kenyon College, Gambier, OH, USA
9.05 1,2,4-Oxadiazines and 1,2,4-Thiadiazines 301
P NORRIS, Youngstown State University, Youngston, OH, USA
9.06 1,2,5-Oxadiazines and 1,2,5-Thiadiazines 345
G W MORROW, University of Dayton, Dayton, OH, USA
9.07 1,2,6-Oxadiazines and 1,2,6-Thiadiazines 355
P M WEINTRAUB, Warren, NJ, USA
9.08 1,3,4-Oxadiazines and 1,3,4-Thiadiazines 401
W-D PFEIFFER, University of Greifswald, Greifswald, Germany
9.09 1,3,5-Oxadiazines and 1,3,5-Thiadiazines 457
N SHOBANA and P FARID, Abbott Laboratories, Abbott Park, 1L, USA
9.10 Dioxazines, Oxathiazines, and Dithiazines 523
E JUARISTI, B R DIAZ, and J L OLIVARES-ROMERO, Centro de Investigation
y de Estudios Avanzados del Instituto Politecnico National, Mexico City, Mexico
9.11 Six-membered Rings with 1,2,4-Oxygen or Sulfur Atoms 569
E KLEINPETER, Universitiit Potsdam, Potsdam, Germany
9.12 1,2,4,5-Tetrazines 641
B STANOVNIK, U GROSELJ, and J SVETE, University of Ljubljana, Ljubljana,
Slovenia
9.13 Other Tetrazines and Pentazines 715
V BENIN, University of Dayton, Dayton, OH, USA
9.14 Other Six-membered Rings with Four or Five Nitrogen, Oxygen, or Sulfur 737
G L FRANCIS, CSIRO, Melbourne, VIC, Australia
9.15 Six-membered Rings with Two or More Heteroatoms with at least One Selenium
or Tellurium 791
F S GUZIEC, Jr. and L J GUZIEC, Southwestern University, Georgetown, TX, USA
9.16 Six-membered Rings with Two or More Heteroatoms with at least One Phosphorus 835
K AFARINKIA, University of Bradford, Bradford, UK
9.17 Six-membered Rings with Two or More Heteroatoms with at least One Arsenic
to Bismuth 875
A GUVEN, Anadolu University, EskiseAir, Turkey
xjv Contents
9.18 Six-mcmbercd Rings with Two or More Heteroatoms with at least One Silicon to Lead 913
I' D LICKISS, Imperial College London, London, UK
9 19 Six-membcred Rings with Two or More Heteroatoms with at least One Boron 961
V D ROMANKNKO, Institute of Bioorganic Chemistry and Petrochemistry, Kiev, Ukraine
J-M SOTIROPOULOS, Universitede Pau et Pays de I'Adour, Pau, France
, . 1009
Index
VOLUME 10 RING SYSTEMS WITH AT LEAST TWO FUSED HETEROGYCLIC
FIVE- OR SIX-MEMBERED RINGS WITH NO BRIDGEHEAD HETEROATOM
10.01 Bicyclic 5-5 Systems: Two Heteroatoms 1:1 1
A KRUTOSIKOVA, University of St. Cyril and Methodius, Trnava, Slovakia
T GRACZA, Slovak University of Technology, Bratislava, Slovakia
10.02 Bicyclic 5-5 Systems: Three Heteroatoms 1:2 65
A J MOORE, University of Sunderland, Sunderland, UK
10.03 Bicyclic 5-5 Systems: Four Heteroatoms 1:3 129
Y A JACKSON and N O TOWNSEND, University of West Indies, Jamaica, West Indies
10.04 Bicyclic 5-5 Systems: Four Heteroatoms 2:2 161
J D WILDEN, University College London, London, UK
10.05 Bicyclic 5-5 Systems: Five Heteroatoms 2:3 and Six Heteroatoms 3:3 189
F HEANEY and L DOYLE, National University of Ireland, Maynooth,
Republic of Ireland
10.06 Bicyclic 5-6 Systems: Two Heteroatoms 1:1 263
A R SHERMAN, College of Notre Dame of Maryland, Baltimore, MD, USA
10.07 Bicyclic 5-6 Systems: Three Heteroatoms 1:2 339
T J DELIA, Central Michigan University, Mt. Pleasant, MI, USA
10.08 Bicyclic 5-6 Systems: Three Heteroatoms 2:1 431
B R BUCKLEY, Loughborough University, Loughborough, UK
10.09 Bicyclic 5-6 Systems: Four Heteroatoms 1:3 493
M C ELLIOTT, Cardiff University, Cardiff, UK
10.10 Bicyclic 5-6 Systems: Four Heteroatoms 3:1 511
B R BUCKLEY and S P NEARY, Loughborough University, Loughborough, UK
10.11 Bicyclic 5-6 Systems: Purines 525
I COLLINS and J J CALDVVELL, The Institute of Cancer Research, Sutton, UK
10.12 Bicyclic 5-6 Systems: Other Four Heteroatoms 2:2 599
M H ELNAGDI, Cairo University, Giza, Egypt
N AL-AWADI, University of Kuwait, Safat, Kuwait
I A ABDELHAMID, Cairo University, Giza, Egypt
10.13 Bicyclic 5-6 Systems: Five Heteroatoms 2:3 or 3:2 661
F ALDABBAGH, National University of Ireland, Galway, Republic of Ireland
10.14 Bicyclic 5-6 Systems: Six and Seven Heteroatoms 703
C A RAMSDEN, Keek University, Keek, UK
10.15 Bicyclic 6-6 Systems: Two Heteroatoms 1:1 713
A P DOBBS, Queen Mary, University of London, London, UK
10.16 Bicyclic 6-6 Systems: Three Heteroatoms 1-2 -jzq
E S H EL ASHRY and N RASHED, Alexandria University, Alexandria, Egypt
Contents xv
10.17 Bicyclic 6-6 Systems: Four Heteroatoms 1:3 847
P W GROUNDWATER and R J ANDERSON, University of Sunderland,
Sunderland, UK
M NYERGES, Technical University of Budapest, Budapest, Hungary
10.18 Bicyclic 6-6 Systems: Pteridines 915
C SUCKLING, G GIBSON, and J HUGGAN, University of Strathclyde, Glasgow, UK
10.19 Bicyclic 6-6 Systems: Other Four Heteroatoms 2:2 977
J M HERBERT, Sanofi-Aventis, Alnwtck, UK
10.20 Bicyclic 6-6 Systems: Five or More Heteroatoms 1093
K HEMMING, University of Huddersfield, Huddersfield, UK
10.21 Tricyclic Systems: Central Carbocyclic Ring with Fused Five-membered Rings 1135
A GRAHAM and M ROBINSON,' University of Wales Swansea, Swansea, UK
10.22 Tricyclic Systems: Central Carbocyclic Ring with Fused Five- and
Six-membered Rings 1201
M P GROZIAK, California State University, East Bay, Hayward, CA, USA
10.23 Tricyclic Systems: Central Carbocyclic Ring with Fused Six-membered Rings 1229
B R BUCKLEY, Loughborough University, Loughborough, UK
Index 1269
VOLUME 11 BICYCLIC 5-5 AND 5-6 FUSED RING SYSTEMS WITH
AT LEAST ONE BRIDGEHEAD (RING JUNCTION) N
11.01 Bicyclic 5-5 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: No
Extra Heteroatom 1
H DHIMANE, UniversitePans Descartes, Pans, France
G LHOMMET, Universite Pierre et Marie Curie-Paris VI, Paris, France
11.02 Bicyclic 5-5 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: One
Extra Heteroatom 1:0 41
J SUFFERT, Universite Louis Pasteur de Strasbourg, Strasbourg, France
11.03 Bicyclic 5-5 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Two
Extra Heteroatoms 2:0 107
L MICOUIN, CNRS, Pans, France
11.04 Bicyclic 5-5 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Two
Extra Heteroatoms 1:1 133
C OLLIVIER, Universite Paul Cezanne-CNRS, Marseille, France
11.05 Bicyclic 5-5 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Three
Extra Heteroatoms 2:1 199
J MARCO-CONTELLES, Instituto de Quimica Orgdnica General (CSIC), Madrid, Spain
E PEREZ-MAYORAL and P BALLESTEROS, UNED, Madrid, Spain
11.06 Bicyclic 5-5 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Three
Extra Heteroatoms 3:0 307
S SABA and J A CIACCIO, Fordham University, Bronx, NY, USA
11.07 Bicyclic 5-5 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Four
Extra Heteroatoms 2:2 325
J ZHU and L NEUVILLE, Institut de Chimie des Substances Naturelles, CNRS,
Gif-sur-Yvette, France
11.08 Bicyclic 5-5 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Four Extra
Heteroatoms 3:1 351
G HILT, W HESS, and C HENGST, Philipps-Universitat Marburg, Marburg, Germany
xvj Contents
11.09 Bicyclic 5-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: No Extra ^
Heteroatom 0:0 .
A BRANDI and S CICCHI, Universita di Firenze, Sesto Fwrentino, bl, Italy
11.10 Bicyclic 5-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: One Extra
Heteroatom 1:0
F COUTY and G EVANO, Universite de Versailles Satnt-Quentm-en-Yvelines, Versailles,
France
11.11 Bicyclic 5-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: One
Extra Heteroatom 0:1 ¦()
M TADDEI, Universita degli Studi di Siena, Siena, Italy
11.12 Bicyciic 5-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Two
Extra Heteroatoms 1:1 ¦'¦''
A C REGAN, University of Manchester, Manchester, UK
11.13 Bicyclic 5-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Two
Extra Heteroatoms 2:0 589
L BISGHOFF, Equipe de Chimie Organique Fine et Heterocyclique (ECOFH), Rouen,
France
11.14 Bicyclic 5-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Two
Extra Heteroatoms 0:2 629
J RODRIGUEZ and T CONSTANTIEUX, Universite Paul Cezanne (Mx-Marseille III),
Marseille, France
11.15 Bicyclic 5-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Three
Extra Heteroatoms 3:0 645
G HAJOS and Z RIEDL, Institute of Biomokcular Chemistry, Chemical Research Center,
Pusztaszeri ut, Hungary
11.16 Bicyclic 5-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Three
Extra Heteroatoms 2:1 671
G HAJOS and Z RIEDL, Institute of Biomokcular Chemistry, Chemical Research Centre,
Budapest, Hungary
11.17 Bicyclic 5-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Three
Extra Heteroatoms 1:2
G HAJOS and Z RIEDL, Institute of Biomokcular Chemistry, Chemical Research Centre,
Budapest, Hungary
11.18 Bicyclic 5-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Four
Extra Heteroatoms 3:1 #19
G HAJOS and Z RIEDL, Institute of Biomokcular Chemistry, Chemical Research Centre,
Budapest, Hungary
11.19 Bicyclic 5-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Four
Extra Heteroatoms 2:2 §47
G HAJOS and Z RIEDL, Institute of Biomokcular Chemistry, Chemical Research Centre
Budapest, Hungary
11.20 Bicyclic 5-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Four
Extra Heteroatoms 1:3 ^y^
G HAJOS and Z RIE DL, Institute of Biomokcular Chemistry, Chemical Research Centre
Budapest, Hungary
11.21 Bicyclic 5-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom- Five
Extra Heteroatoms 3:2 909
G HAJOS and Z RIEDL, Institute of Biomokcular Chemistry, Chemical Research Centre
Budapest, Hungary
Index
919
Contents xvii
VOLUME 12 FIVE- AND SIX-MEMBERED FUSED SYSTEMS WITH
BRIDGEHEAD (RING JUNCTION) HETEROATOMS CONCLUDED: 6-6
BICYCLIC WITH ONE OR TWO N OR OTHER HETEROATOMS;
POLYCYCLIC; SPIROCYCLIC
12.01 Bicyclic 6-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: No Extra
Heteroatom 1
C AVENDANO and J C MENENDEZ, Universidad Complutense, Madrid, Spain
12.02 Bicyclic 6-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: One
Extra Heteroatom 1:0 77
I HERMECZ and L VASVARI-DEBRECZY, Chinoin Pharmaceutical and Chemical
Works Ltd., Budapest, Hungary
12.03 Bicyclic 6-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Two
Extra Heteroatoms 2:0 219
P MATYUS and P TAPOLCSANYI, Semmelweis University, Budapest, Hungary
12.04 Bicyclic 6-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Two
Extra Heteroatoms 1:1 257
I HERMECZ and L VASVARI-DEBRECZY, Chinoin Pharmaceutical and Chemical
Works Ltd., Budapest, Hungary
12.05 Bicyclic 6-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Three
Extra Heteroatoms 3:0 321
M P MAHAJAN and C MOHAN, Guru Nanak Dev University, Amritsar, India
12.06 Bicyclic 6-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Three
Extra Heteroatoms 2:1 327
M P MAHAJAN, G BHARGAVA, and C MOHAN, Guru Nanak Dev University,
Amritsar, India
12.07 Bicyclic 6-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Four
Extra Heteroatoms 3:1 341
M P MAHAJAN and C MOHAN, Guru Nanak Dev University, Amritsar, India
12.08 Bicyclic 6-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Four
Extra Heteroatoms 2:2 347
M P MAHAJAN, A MARWAHA, and C MOHAN, Guru Nanak Dev University,
Amritsar, India
12.09 Bicyclic 6-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Five
Extra Heteroatoms 3:2 357
M P MAHAJAN and C MOHAN, Guru Nanak Dev University, Amritsar, India
12.10 Bicyclic Systems with Two Bridgehead (Ring Junction) Nitrogen Atoms 365
S RADL, Zentiva - Research Institute for Pharmacy and Biochemistry, Prague,
Czech Republic
12.11 Bicyclic Systems with Bridgehead (Ring Junction) Sulfur, Selenium,
or Tellurium Atoms 481
I FORRISTAL, King Fahd University of Petroleum Minerals, Dhahran, Saudi Arabia
12.12 Bicyclic Systems with Bridgehead (Ring Junction) Phosphorus, Arsenic,
Antimony, or Bismuth Atoms 527
S SCHWIKKARD, Kingston University, Kingston, UK
12.13 Bicyclic Systems with Bridgehead (Ring Junction) Boron Atoms 573
Yu N BUBNOV, M E GURSKII, and S Yu ERDYAKOV, Russian Academy of
Sciences, Moscow, Russia
12.14 Three Heterocyclic Rings Fused (5-5-5) 635
K C MAJUMDAR and S K CHATTOPADHYAY, University of Kalyani, Kalyani, India
xviii Contents
12.15 Three Heterocyclic Rings Fused (5-6-5)
S HILTON, The Institute of Cancer Research, Sutton, UK
S ROSSITER, University of Hertfordshire, Hatfield, UK
12.16 Three Heterocyclic Rings Fused (5-5-6)
R L RIGGS, BASF AG, Ludwigshafen, Germany
D M SMITH, University of St Andrews, St Andrews, UK
12.17 Three Heterocyclic Rings Fused (5-6-6) 857
R L RIGGS, BASF AG, Ludwigshafen, Germany
D M SMITH, University of St. Andrews, St. Andrews, UK
12.18 Three Heterocyclic Rings Fused (6-5-6) 975
L STRFKOWSKI, J SACZEWSKI, and M HENARY, Georgia State University,
Atlanta, GA, USA
12.19 Three Heterocyclic Rings Fused (6-6-6) 1007
L STREKOWSKI, M HENARY, and M MOJZYCH, Georgia State University,
Atlanta, GA, USA
12.20 Systems with a Spirocyclic Heteroatom 1037
N M AHMAD, The Institute of Cancer Research, Sutton, UK
\Z.Z\ Compounds containing a Spiro Phosphorus Atom 1065
N A WILLIAMS, Kingston University, Kingston upon Thames, UK
Index 1127
VOLUME 13 SEVEN-MEMBERED HETEROCYCLIC RINGS AND THEIR FUSED
DERIVATIVES
13.01 Azepines and their Fused-ring Derivatives 1
J B BREMNER, University of Wollongong, Wollongong, NSW, Australia
S SAMOSORN, Srinakharinwirot University, Bangkok, Thailand
13.02 Oxepanes and Oxepines 45
L I BELEN'KII, Russian Academy of Sciences, Moscow, Russia
13.03 Thiepanes and Thiepines 97
S YAMAZAKI, Nara University of Education, Nara, Japan
13.04 1,2-Diazepines 143
T P MEAGHER, TEKA Consulting, Indianapolis, IN, USA
R MURUGAN, Vertellus Specialties Inc, Indianapolis, IN, USA
13.05 1,3-Diazepines j^j
W M DE BORGGRAEVE and A M VAN DEN BOGAERT, K ULeuven,
I*liven, Belgium
13.06 1,4-Diazepines jg-^
N A MEANWELL and M A WALKER, Bristol-Myers Squibb Research and
Development, Wallingford, CT, USA
13.07 1,2-Oxazepines and 1,2-Thiazepines ?37
J B BREMNER, University of Wollongong, Wollongong, NSW, Australia
S SAMOSORN, Srinakharinwirot University, Bangkok, Thailand
13.08 1,3-Oxazepines and 1,3-Thiazepines 245
Jc \ *ISScI^ER' University °f Wollongong, Wollongong, NSW, Australia
b SAMOSORN, Snnakhartnwirot University, Bangkok, Thailand
13.09 1,4-Oxazepines and 1,4-Thiazepines 2SS
W DEHAEN and T H NGO, University of Leuven, Leuven, Belgium
Contents xix
13.10 1,2-Dioxepanes, 1,2-Oxathiepanes, and 1,2-Dithiepanes 299
M J HADDADIN and C J NACHEF, American University of Beirut, Beirut,
Lebanon
13.11 1,3-Dioxepanes, 1,3-Oxathiepanes, and 1,3-Dithiepanes 321
H FRAUENRATH and S FLOCK, University of Kassel, Kassel, Germany
13.12 1,4-Dioxepanes, 1,4-Oxathiepanes, and 1,4-Dithiepanes 367
H FRAUENRATH and S FLOCK, Universitat GH Kassel, Kassel, Germany
R MURUGAN, Vertellus Specialties Inc., Indianapolis, IN, USA
E F V SCRIVEN, University of Florida, Gainesville, FL, USA
13.13 Seven-membered Rings with Three Heteroatoms 1,2,3 387
A KISELYOV and A KHVAT, ChemDw Inc., San Diego, CA, USA
13.14 Seven-membered Rings with Three Heteroatoms 1,2,4 399
G I YRANZO and E L MOYANO, Universidad Nacwnal de Cordoba, Cordoba,
Argentina
13.15 Seven-membered Rings with Three Heteroatoms 1,2,5 433
R RANJITH KUMAR and S PERUMAL, Madurai Kamaraj University,
Madurai, India
M BALASUBRAMANIAN, Pfizer, Inc., Groton, CT, USA
13.16 Seven-membered Rings with Three Heteroatoms 1,3,5 489
0 V DENISKO, Chemical Abstracts Service, Columbus, OH, USA
13.17 Seven-membered Rings with Four or More Heteroatoms 529
G N NIKONOV, Alchem Laboratories Co., Alachua, FL, USA
Index 571
VOLUME 14 EIGHT-MEMBERED AND LARGER HETEROCYGLIC RINGS
AND THEIR FUSED DERIVATIVES, OTHER SEVEN-MEMBERED RINGS
14.01 Eight-membered Rings with One Nitrogen Atom 1
D C ONICIU, University of Florida, Gainesville, FL, USA
14.02 Eight-membered Rings with One Oxygen Atom 49
A M S SILVA and A C TOME, University of Aveiro, Aveiro, Portugal
14.03 Eight-membered Rings with One Sulfur Atom 89
H ECKERT, Technical University of Munich, Garching, Germany
14.04 Eight-membered Rings with Two Heteroatoms 1,2 99
G CIRRINCIONE and P DIANA, Universitd degli Studi di Palermo, Palermo, Italy
14.05 Eight-membered Rings with Two Heteroatoms 1,3 169
G CIRRINCIONE and P DIANA, Universitd degli Studi di Palermo, Palermo, Italy
14.06 Eight-membered Rings with Two Heteroatoms 1,4 255
1 SHCHERBAKOVA, MediProPharma, Inc., Midvale, (IT, USA
14.07 Eight-membered Rings with Two Heteroatoms 1,5 303
G CIRRINCIONE and P DIANA, Universitd degli Studi di Palermo, Palermo, Italy
14.08 Eight-membered Rings with Three Heteroatoms 475
D O TYMOSHENKO, Albany Molecular Research, Inc., Albany, NY, USA
14.09 Eight-membered Rings with Four or More Heteroatoms 517
I SHCHERBAKOVA, MediProPharma, Inc., Midvale, UT, USA
14.10 Nine-membered Rings 547
D O TYMOSHENKO, AMRI, Albany, NY, USA
xx Contents
14.11 Ten-membered Rings or Larger with One or More Nitrogen Atoms 613
P HERMANN and J KOTEK, Universita Karlova, Prague, Czech Republic
14.12 Ten-membered Rings or Larger with One or More Oxygen Atoms 667
S PAPPALARDO, Universita di Catania, Catania, Italy
M F PARISI, Universita di Messina, Messina, Italy
14.13 Ten-membered Rings or Larger with One or More Sulfur Atoms 751
H ECKERT, Technical University of Munich, Garching, Germany
M ROLLER, Bundeswehr Institute of Pharmacology and Toxicology, Munich, Germany
14.14 Ten-membered Rings or Larger with One or More Nitrogen and Oxygen
and/or Sulfur Atoms 803
G W GOKEL and E K ELLIOTT, Washington University School of Medicine,
St. Louis, MO, USA
14.15 Ten-membered Rings or Larger with One or More Oxygen and Sulfur Atoms 829
Y HABATA, Toho University, Chiba, Japan
14.16 Rings containing Selenium or Tellurium 863
G L SOMMEN, Lonza AG, Walliser Werke, Visp, Switzerland
14.17 Rings containing Phosphorus 901
A M SHESTOPALOV, Zelinsky Institute of Organic Chemistry, Moscow, Russia
A A SHESTOPALOV, Duke University, Durham, NC, USA '
14.18 Rings containing Arsenic, Antimony, or Bismuth 945
V D ROMANENKO, Institute of Bioorganic Chemistry and Petrochemistry, Kiev, Ukraine
J-M SOTIROPOULOS, Universite de Pau et Pays de I'Adour, Pau, France
14.19 Rings containing Silicon to Lead 979
F SACZEWSKI and A KORNICKA, Medical University of Gdansk, Gdansk, Poland
14.20 Rings containing Boron 10}9
G \V MORROW, University of Dayton, Dayton, OH, USA
14.21 Rings containing Other Elements 1051
T P MEAGHER, TEKA Consulting, Indianapolis, IN, USA
14.22 Multiple Macroheterocyclic Rings 1071
A M-P PEDERSON and H W GIBSON, Virginia Polytechnic Institute and State
University, Blacksburg, VA, USA
Indt"X 1087
VOLUME 15 CUMULATIVE SUBJECT INDEX !
.«*
'«?'
Introduction
Alan R. Katritzky, Christopher A. Ramsden, Eric F. V. Scriven, and Richard J. K. Taylor
1 Scope, Significance, and Aims 50
1.1 Scope 50
1.2 Significance 50
1.3 Aims of CHEC-I, CHEC-II and CHEC-III 50
2 Arrangement of the Work in Volumes 51
2.1 Relationship of CHEC-III to CHEC-I and CHEC-II 51
2.2 Arrangement of CHEC-III in Volumes 51
2.3 Arrangement of CHEC-II in Volumes 51
2.4 Arrangement of CHEC-I in Volumes 52
3 Rationale for Arrangement of Material in Individual Volumes 52
3.1 Major Divisions of Carbocyclic and Heterocyclic Chemistry 52
3.2 Saturated Heterocyclic Compounds 53
3.3 Partially Unsaturated Heterocyclic Compounds 53
3.4 Heteroaromatic Compounds 53
3.5 Characteristics of Heteroatoms in Rings 53
3.6 The General Chapters of CHEC-I 54
4 Organization of Individual Monograph Chapters 54
4.1 Introduction 55
4.2 Theoretical Methods 55
4.3 Experimental Structural Methods 55
4.4 Thermodynamic Aspects 55
4.5 Reactivity of Fully Conjugated Rings 55
4.6 Reactivity of Nonconjugated Rings 56
4.7 Reactivity of Substituents Attached to Ring Carbon Atoms 56
4.8 Reactivity of Substituents Attached to Ring Heteroatoms 56
4.9 Ring Syntheses Classified by Number of Ring Atoms in Each Component 56
4.10 Ring Synthesis by Transformation of Another Ring 56
4.11 Synthesis of Particular Classes of Compounds and Critical Comparison of the Various
Routes Available 56
4.12 Important Compounds and Applications 56
5 The Reference System 56
6 The Indexes 57
6.1 Ring Index 57
6.2 Subject Index 57 |
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spelling | Comprehensive heterocyclic chemistry III [a review of the literature 1995 - 2007] 15 Cumulative subject index execut.-ed. Alan R. Katritzky. Eds-in-chief Christopher A. Ramsden ... 1. ed. Amsterdam [u.a.] Elsevier 2008 LIX, 350 S. Ill. txt rdacontent n rdamedia nc rdacarrier Katritzky, Alan R. 1928-2014 Sonstige (DE-588)137133421 oth Ramsden, Christopher A. Sonstige oth (DE-604)BV023477408 15 HBZ Datenaustausch application/pdf http://bvbr.bib-bvb.de:8991/F?func=service&doc_library=BVB01&local_base=BVB01&doc_number=016660028&sequence=000002&line_number=0001&func_code=DB_RECORDS&service_type=MEDIA Inhaltsverzeichnis |
spellingShingle | Comprehensive heterocyclic chemistry III [a review of the literature 1995 - 2007] |
title | Comprehensive heterocyclic chemistry III [a review of the literature 1995 - 2007] |
title_auth | Comprehensive heterocyclic chemistry III [a review of the literature 1995 - 2007] |
title_exact_search | Comprehensive heterocyclic chemistry III [a review of the literature 1995 - 2007] |
title_exact_search_txtP | Comprehensive heterocyclic chemistry III [a review of the literature 1995 - 2007] |
title_full | Comprehensive heterocyclic chemistry III [a review of the literature 1995 - 2007] 15 Cumulative subject index execut.-ed. Alan R. Katritzky. Eds-in-chief Christopher A. Ramsden ... |
title_fullStr | Comprehensive heterocyclic chemistry III [a review of the literature 1995 - 2007] 15 Cumulative subject index execut.-ed. Alan R. Katritzky. Eds-in-chief Christopher A. Ramsden ... |
title_full_unstemmed | Comprehensive heterocyclic chemistry III [a review of the literature 1995 - 2007] 15 Cumulative subject index execut.-ed. Alan R. Katritzky. Eds-in-chief Christopher A. Ramsden ... |
title_short | Comprehensive heterocyclic chemistry III |
title_sort | comprehensive heterocyclic chemistry iii a review of the literature 1995 2007 cumulative subject index |
title_sub | [a review of the literature 1995 - 2007] |
url | http://bvbr.bib-bvb.de:8991/F?func=service&doc_library=BVB01&local_base=BVB01&doc_number=016660028&sequence=000002&line_number=0001&func_code=DB_RECORDS&service_type=MEDIA |
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