Handbook of preformulation: chemical, biological, and botanical drugs
Gespeichert in:
1. Verfasser: | |
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Format: | Buch |
Sprache: | English |
Veröffentlicht: |
New York [u.a.]
Informa Healthcare
2007
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Schlagworte: | |
Online-Zugang: | Publisher description Inhaltsverzeichnis |
Beschreibung: | Includes bibliographical references and index |
Beschreibung: | xix, 446 p. Ill., graph. Darst. 24 cm |
ISBN: | 0849371937 9780849371936 |
Internformat
MARC
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100 | 1 | |a Niazi, Sarfaraz Khan |d 1949- |e Verfasser |0 (DE-588)133089851 |4 aut | |
245 | 1 | 0 | |a Handbook of preformulation |b chemical, biological, and botanical drugs |c Sarfaraz K. Niazi |
264 | 1 | |a New York [u.a.] |b Informa Healthcare |c 2007 | |
300 | |a xix, 446 p. |b Ill., graph. Darst. |c 24 cm | ||
336 | |b txt |2 rdacontent | ||
337 | |b n |2 rdamedia | ||
338 | |b nc |2 rdacarrier | ||
500 | |a Includes bibliographical references and index | ||
650 | 4 | |a Médicaments - Formes pharmaceutiques - Guides, manuels, etc | |
650 | 4 | |a Mélange - Guides, manuels, etc | |
650 | 4 | |a Techniques pharmaceutiques - Guides, manuels, etc | |
650 | 4 | |a Pharmaceutical technology |v Handbooks, manuals, etc | |
650 | 4 | |a Mixing |v Handbooks, manuals, etc | |
650 | 4 | |a Drugs |x Dosage forms |v Handbooks, manuals, etc | |
650 | 4 | |a Chemistry, Pharmaceutical |x methods |v Handbooks | |
650 | 4 | |a Chemistry, Physical |x methods |v Handbooks | |
650 | 4 | |a Dosage Forms |v Handbooks | |
650 | 4 | |a Drug Stability |v Handbooks | |
856 | 4 | |u http://www.loc.gov/catdir/enhancements/fy0661/2006046566-d.html |3 Publisher description | |
856 | 4 | 2 | |m GBV Datenaustausch |q application/pdf |u http://bvbr.bib-bvb.de:8991/F?func=service&doc_library=BVB01&local_base=BVB01&doc_number=016148608&sequence=000001&line_number=0001&func_code=DB_RECORDS&service_type=MEDIA |3 Inhaltsverzeichnis |
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Datensatz im Suchindex
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adam_text | HANDBOOK OF PREFORMULATION LNEMICAL, MOLOGICAL, AND DOLANICAL JJRUGS
SARFARAZ K. NIAZI PHARMACEUTICAL SCIENTIST INC. DEERFIELD, ILLINOIS,
U.S.A. INFORMA HEALTHCARE NEW YORK LONDON CONTENTS PREFACE . . . . V
LIST OF APPENDICES, FIGURES, SCHEMES, AND TABLES .... XIII 1. DRUG
DISCOVERY TRENDS / INTRODUCTION .... / DEVELOPMENT PHASES .... 2 PRODUCT
LIFE CYCLE .... 6 NEW PATHWAYS TO DISCOVERY .... // REFERENCES .... 23
BIBLIOGRAPHY .... 23 Z. INTELLECTUAL PROPERTY CONSIDERATIONS 33
INTRODUCTION .... 33 PATENTING STRATEGIES .... 33 PATENTING SYSTEMS ....
35 WHAT IS A PATENT? .... 35 PATENT MYTHS .... 36 WHAT IS NOT
PATENTABLE? 38 PATENT SEARCH .... 38 COMPONENTS OF A PATENT APPLICATION
.... 44 UNDERSTANDING CLAIMS .... 49 FOOD AND DRUG ADMINISTRATION ....
55 REFERENCES .... 56 BIBLIOGRAPHY .... 56 I. THE SCOPE OF
PREFORMULATION STUDIES 57 INTRODUCTION .... 57 PREFORMULATION TESTING
CRITERIA .... 57 REGULATORY REQUIREMENTS .... 58 TESTING SYSTEMS .... 65
SOLID-STATE CHARACTERIZATION .... 69 TRANSPORT ACROSS BIOLOGICAL
MEMBRANES .... 77 REFERENCES .... 79 BIBLIOGRAPHY .... 79 4.
DISSOCIATION, PARTITIONING, AND SOLUBILITY 87 INTRODUCTION .... 87 THE
IONIZATION PRINCIPLE .... 87 QUANTITATIVE STRUCTURE-ACTIVITY
RELATIONSHIPS .... 98 PARTITIONING .... 105 MEASUREMENT STRATEGIES ....
113 REFERENCES .... 122 BIBLIOGRAPHY .... 122 APPENDIX 1 .... 131 XVII
CONTENTS 5. RELEASE, DISSOLUTION, AND PERMEATION 141 INTRODUCTION ....
141 RELEASE .... 141 ASSAY SYSTEMS .... 147 THE BIOPHARMACEUTICS DRUG
CLASSIFICATION SYSTEMS .... 156 REFERENCES . ... 159 BIBLIOGRAPHY ...
159 APPENDIX 1 .... 168 6. SOLID-STATE PROPERTIES 197 INTRODUCTION ....
197 CRYSTAL MORPHOLOGY ... 197 POLYMORPHISM .... 203 HIGH-THROUGHPUT
CRYSTAL SCREENING .... 207 SOLVATES .... 210 HYDRATES .... 210 AMORPHOUS
FORMS .... 212 HYGROSCOPICITY .... 212 SOLUBILITY 213 STUDY METHODS ....
218 REFERENCES .... 231 BIBLIOGRAPHY .... 231 7. DOSAGE FORM
CONSIDERATIONS IN PREFORMULATION 241 INTRODUCTION .... 241 SOLID DOSAGE
FORM CONSIDERATIONS .... 241 SOLUTION FORMULATIONS .... 262 EMULSION
FORMULATIONS .... 26_? FREEZE-DRIED FORMULATIONS .... 271 SUSPENSIONS
.... 272 TOPICAL 273 PULMONARY DELIVERY .... 274 GENERAL COMPATIBILITY
.... 275 REFERENCES .... 275 BIBLIOGRAPHY .... 276 8. CHEMICAL DRUG
SUBSTANCE CHARACTERIZATION 287 INTRODUCTION .... 287 SCHEME OF
CHARACTERIZATION .... 288 IMPURITIES ?/7 GOOD MANUFACTURING PRACTICE
.... 322 REFERENCES .... 326 BIBLIOGRAPHY .... 326 9. CHARACTERIZATION
OF BIOPHARMACEUTICAL DRUGS 329 INTRODUCTION .... 329 PREFORMULATION
STUDIES .... 333 PACKAGING AND MATERIALS .... 348 PHYSIO-CHEMICAL
CHARACTERIZATION TESTS .... 385 DESIGN OF PREFORMULATION STUDIES ....
387 REFERENCES .... 388 BIBLIOGRAPHY .... 388 1O. CHARACTERIZATION OF
PHYTOMEDICINES 391 INTRODUCTION .... 391 REGULATORY STATUS .... 392
CONTENTS XIX CHARACTERISTICS OF PHYTOMEDICINES .... 392 EFFICACY AND
SAFETY .... 399 REGULATORY FILING PROCEDURE .... 400 STARTING MATERIAL
.... 403 STABILITY TESTING .... 406 BIBLIOGRAPHY .... 410 GLOSSARY OF
TERMS .... 429 INDEX 432
|
adam_txt |
HANDBOOK OF PREFORMULATION LNEMICAL, MOLOGICAL, AND DOLANICAL JJRUGS
SARFARAZ K. NIAZI PHARMACEUTICAL SCIENTIST INC. DEERFIELD, ILLINOIS,
U.S.A. INFORMA HEALTHCARE NEW YORK LONDON CONTENTS PREFACE . . . . V
LIST OF APPENDICES, FIGURES, SCHEMES, AND TABLES . XIII 1. DRUG
DISCOVERY TRENDS / INTRODUCTION . / DEVELOPMENT PHASES . 2 PRODUCT
LIFE CYCLE . 6 NEW PATHWAYS TO DISCOVERY . // REFERENCES . 23
BIBLIOGRAPHY . 23 Z. INTELLECTUAL PROPERTY CONSIDERATIONS 33
INTRODUCTION . 33 PATENTING STRATEGIES . 33 PATENTING SYSTEMS .
35 WHAT IS A PATENT? . 35 PATENT MYTHS . 36 WHAT IS NOT
PATENTABLE? 38 PATENT SEARCH . 38 COMPONENTS OF A PATENT APPLICATION
. 44 UNDERSTANDING CLAIMS . 49 FOOD AND DRUG ADMINISTRATION .
55 REFERENCES . 56 BIBLIOGRAPHY . 56 I. THE SCOPE OF
PREFORMULATION STUDIES 57 INTRODUCTION . 57 PREFORMULATION TESTING
CRITERIA . 57 REGULATORY REQUIREMENTS . 58 TESTING SYSTEMS . 65
SOLID-STATE CHARACTERIZATION . 69 TRANSPORT ACROSS BIOLOGICAL
MEMBRANES . 77 REFERENCES . 79 BIBLIOGRAPHY . 79 4.
DISSOCIATION, PARTITIONING, AND SOLUBILITY 87 INTRODUCTION . 87 THE
IONIZATION PRINCIPLE . 87 QUANTITATIVE STRUCTURE-ACTIVITY
RELATIONSHIPS . 98 PARTITIONING . 105 MEASUREMENT STRATEGIES .
113 REFERENCES . 122 BIBLIOGRAPHY . 122 APPENDIX 1 . 131 XVII
CONTENTS 5. RELEASE, DISSOLUTION, AND PERMEATION 141 INTRODUCTION .
141 RELEASE . 141 ASSAY SYSTEMS . 147 THE BIOPHARMACEUTICS DRUG
CLASSIFICATION SYSTEMS . 156 REFERENCES . . 159 BIBLIOGRAPHY .
159 APPENDIX 1 . 168 6. SOLID-STATE PROPERTIES 197 INTRODUCTION .
197 CRYSTAL MORPHOLOGY . 197 POLYMORPHISM . 203 HIGH-THROUGHPUT
CRYSTAL SCREENING . 207 SOLVATES . 210 HYDRATES . 210 AMORPHOUS
FORMS . 212 HYGROSCOPICITY . 212 SOLUBILITY 213 STUDY METHODS .
218 REFERENCES . 231 BIBLIOGRAPHY . 231 7. DOSAGE FORM
CONSIDERATIONS IN PREFORMULATION 241 INTRODUCTION . 241 SOLID DOSAGE
FORM CONSIDERATIONS . 241 SOLUTION FORMULATIONS . 262 EMULSION
FORMULATIONS . 26_? FREEZE-DRIED FORMULATIONS . 271 SUSPENSIONS
. 272 TOPICAL 273 PULMONARY DELIVERY . 274 GENERAL COMPATIBILITY
. 275 REFERENCES . 275 BIBLIOGRAPHY . 276 8. CHEMICAL DRUG
SUBSTANCE CHARACTERIZATION 287 INTRODUCTION . 287 SCHEME OF
CHARACTERIZATION . 288 IMPURITIES ?/7 GOOD MANUFACTURING PRACTICE
. 322 REFERENCES . 326 BIBLIOGRAPHY . 326 9. CHARACTERIZATION
OF BIOPHARMACEUTICAL DRUGS 329 INTRODUCTION . 329 PREFORMULATION
STUDIES . 333 PACKAGING AND MATERIALS . 348 PHYSIO-CHEMICAL
CHARACTERIZATION TESTS . 385 DESIGN OF PREFORMULATION STUDIES .
387 REFERENCES . 388 BIBLIOGRAPHY . 388 1O. CHARACTERIZATION OF
PHYTOMEDICINES 391 INTRODUCTION . 391 REGULATORY STATUS . 392
CONTENTS XIX CHARACTERISTICS OF PHYTOMEDICINES . 392 EFFICACY AND
SAFETY . 399 REGULATORY FILING PROCEDURE . 400 STARTING MATERIAL
. 403 STABILITY TESTING . 406 BIBLIOGRAPHY . 410 GLOSSARY OF
TERMS . 429 INDEX 432 |
any_adam_object | 1 |
any_adam_object_boolean | 1 |
author | Niazi, Sarfaraz Khan 1949- |
author_GND | (DE-588)133089851 |
author_facet | Niazi, Sarfaraz Khan 1949- |
author_role | aut |
author_sort | Niazi, Sarfaraz Khan 1949- |
author_variant | s k n sk skn |
building | Verbundindex |
bvnumber | BV022944008 |
callnumber-first | R - Medicine |
callnumber-label | RS199 |
callnumber-raw | RS199.F67 |
callnumber-search | RS199.F67 |
callnumber-sort | RS 3199 F67 |
callnumber-subject | RS - Pharmacy |
classification_rvk | VX 5200 |
ctrlnum | (OCoLC)70218023 (DE-599)BVBBV022944008 |
dewey-full | 615/.19 |
dewey-hundreds | 600 - Technology (Applied sciences) |
dewey-ones | 615 - Pharmacology and therapeutics |
dewey-raw | 615/.19 |
dewey-search | 615/.19 |
dewey-sort | 3615 219 |
dewey-tens | 610 - Medicine and health |
discipline | Chemie / Pharmazie Medizin |
discipline_str_mv | Chemie / Pharmazie Medizin |
format | Book |
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id | DE-604.BV022944008 |
illustrated | Illustrated |
index_date | 2024-07-02T18:59:06Z |
indexdate | 2024-07-09T21:08:14Z |
institution | BVB |
isbn | 0849371937 9780849371936 |
language | English |
lccn | 2006046566 |
oai_aleph_id | oai:aleph.bib-bvb.de:BVB01-016148608 |
oclc_num | 70218023 |
open_access_boolean | |
owner | DE-19 DE-BY-UBM |
owner_facet | DE-19 DE-BY-UBM |
physical | xix, 446 p. Ill., graph. Darst. 24 cm |
publishDate | 2007 |
publishDateSearch | 2007 |
publishDateSort | 2007 |
publisher | Informa Healthcare |
record_format | marc |
spelling | Niazi, Sarfaraz Khan 1949- Verfasser (DE-588)133089851 aut Handbook of preformulation chemical, biological, and botanical drugs Sarfaraz K. Niazi New York [u.a.] Informa Healthcare 2007 xix, 446 p. Ill., graph. Darst. 24 cm txt rdacontent n rdamedia nc rdacarrier Includes bibliographical references and index Médicaments - Formes pharmaceutiques - Guides, manuels, etc Mélange - Guides, manuels, etc Techniques pharmaceutiques - Guides, manuels, etc Pharmaceutical technology Handbooks, manuals, etc Mixing Handbooks, manuals, etc Drugs Dosage forms Handbooks, manuals, etc Chemistry, Pharmaceutical methods Handbooks Chemistry, Physical methods Handbooks Dosage Forms Handbooks Drug Stability Handbooks http://www.loc.gov/catdir/enhancements/fy0661/2006046566-d.html Publisher description GBV Datenaustausch application/pdf http://bvbr.bib-bvb.de:8991/F?func=service&doc_library=BVB01&local_base=BVB01&doc_number=016148608&sequence=000001&line_number=0001&func_code=DB_RECORDS&service_type=MEDIA Inhaltsverzeichnis |
spellingShingle | Niazi, Sarfaraz Khan 1949- Handbook of preformulation chemical, biological, and botanical drugs Médicaments - Formes pharmaceutiques - Guides, manuels, etc Mélange - Guides, manuels, etc Techniques pharmaceutiques - Guides, manuels, etc Pharmaceutical technology Handbooks, manuals, etc Mixing Handbooks, manuals, etc Drugs Dosage forms Handbooks, manuals, etc Chemistry, Pharmaceutical methods Handbooks Chemistry, Physical methods Handbooks Dosage Forms Handbooks Drug Stability Handbooks |
title | Handbook of preformulation chemical, biological, and botanical drugs |
title_auth | Handbook of preformulation chemical, biological, and botanical drugs |
title_exact_search | Handbook of preformulation chemical, biological, and botanical drugs |
title_exact_search_txtP | Handbook of preformulation chemical, biological, and botanical drugs |
title_full | Handbook of preformulation chemical, biological, and botanical drugs Sarfaraz K. Niazi |
title_fullStr | Handbook of preformulation chemical, biological, and botanical drugs Sarfaraz K. Niazi |
title_full_unstemmed | Handbook of preformulation chemical, biological, and botanical drugs Sarfaraz K. Niazi |
title_short | Handbook of preformulation |
title_sort | handbook of preformulation chemical biological and botanical drugs |
title_sub | chemical, biological, and botanical drugs |
topic | Médicaments - Formes pharmaceutiques - Guides, manuels, etc Mélange - Guides, manuels, etc Techniques pharmaceutiques - Guides, manuels, etc Pharmaceutical technology Handbooks, manuals, etc Mixing Handbooks, manuals, etc Drugs Dosage forms Handbooks, manuals, etc Chemistry, Pharmaceutical methods Handbooks Chemistry, Physical methods Handbooks Dosage Forms Handbooks Drug Stability Handbooks |
topic_facet | Médicaments - Formes pharmaceutiques - Guides, manuels, etc Mélange - Guides, manuels, etc Techniques pharmaceutiques - Guides, manuels, etc Pharmaceutical technology Handbooks, manuals, etc Mixing Handbooks, manuals, etc Drugs Dosage forms Handbooks, manuals, etc Chemistry, Pharmaceutical methods Handbooks Chemistry, Physical methods Handbooks Dosage Forms Handbooks Drug Stability Handbooks |
url | http://www.loc.gov/catdir/enhancements/fy0661/2006046566-d.html http://bvbr.bib-bvb.de:8991/F?func=service&doc_library=BVB01&local_base=BVB01&doc_number=016148608&sequence=000001&line_number=0001&func_code=DB_RECORDS&service_type=MEDIA |
work_keys_str_mv | AT niazisarfarazkhan handbookofpreformulationchemicalbiologicalandbotanicaldrugs |