Medicinal chemistry for the 21st century:
Gespeichert in:
Format: | Buch |
---|---|
Sprache: | English |
Veröffentlicht: |
Oxford u.a.
Blackwell Scientific Publ.
1992
|
Ausgabe: | 1. publ. |
Schriftenreihe: | A "Chemistry for the 21st century" monograph
|
Schlagworte: | |
Online-Zugang: | Inhaltsverzeichnis |
Beschreibung: | XII, 402 S. Ill., graph. Darst. |
ISBN: | 0632034084 |
Internformat
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245 | 1 | 0 | |a Medicinal chemistry for the 21st century |c International Union of Pure and Applied Chemistry. Ed. by C. G. Wermuth |
250 | |a 1. publ. | ||
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650 | 4 | |a Chemistry, Pharmaceutical |x trends | |
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Datensatz im Suchindex
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adam_text | INTERNATIONAL UNION OF PURE AND APPLIED CHEMISTRY MEDICINAL CHEMISTRY
FOR THE 21ST CENTURY IUPAC A CHEMISTRY FOR THE 21ST CENTURY MONOGRAPH
EDITED BY C.G. WERMUTH LABORATOIRE DE PHARMACOCHIMIE MOLECULAIRE FACULTE
DE PHARMACIE UNIVERSITE LOUIS PASTEUR STRASBOURG FRANCE WITH N. KOGA
DAIICHI PHARMACEUTICAL CO., LTD TOKYO 103 JAPAN H. KONIG BASF
AKTIENGESELISCHAFT D-6700 LUDWIGSHAFEN GERMANY B.W. METCALF SMITHKLINE
BEECHAM PHARMACEUTICALS KING OF PRUSSIA, PA 19406-2799 USA OXFORD
BLACKWELL SCIENTIFIC PUBLICATIONS LONDON EDINBURGH BOSTON MELBOURNE
PARIS BERLIN VIENNA CONTENTS CONTRIBUTORS IX PREFACE XI PART 1: NEW LEAD
DISCOVERY HISTORICAL PERSPECTIVES 1 PAST APPROACHES TO DISCOVERING NEW
DRUGS 3 C.R. GANELLIN 2 REFLECTIONS AND PERSPECTIVES 13 P.A.J. JANSSEN
AND J.P. TOLLENAERE STRATEGIES FOR THE CREATION OF NEW DRUGS 3 TRENDS IN
NEW LEAD IDENTIFICATION: A STRUCTURAL APPROACH 25 J.H. MUSSER 4 FROM
MEMBRANE TO GENOMIC PHARMACOLOGY OR FROM SHORT-TERM TO LONG-TERM EFFECTS
39 P.M. LADURON 5 FUTURE APPLICATIONS OF OLIGONUCLEOTIDES IN ANTIVIRAL
AND ANTITUMORAL CHEMOTHERAPY 45 P. HERDEWIJN AND E. DE CLERCQ PART 2:
PROTEIN STRUCTURE-FUNCTION RELATIONSHIPS CLONING AND STRUCTURAL STUDIES
ON RECEPTORS AND ENZYMES 6 MOLECULAR BIOLOGY OF DRUG RECEPTORS AND THE
ADVENT OF REVERSE PHARMACOLOGY 63 J.-C. SCHWARTZ 7 A STRUCTURAL BASIS
FOR PROTEINASE-PROTEIN INHIBITOR INTERACTION 73 W. BODE AND R. HUBER
DETECTION OF NEW ENZYMES AND RECEPTORS BY HYBRIDIZATION TECHNIQUE 8 NEW
APPROACHES TO ISOLATION, EXPRESSION AND MOLECULAR MODELLING OF PROTEASES
107 J.H. MCKERROW, F.E. COHEN, C.S. CRAIK AND J.A. SAKANARI VI CONTENTS
9 NEW ERA OF BIOCHEMISTRY: CYTOKINE SIGNAL NETWORK AND ITS IMPLICATION
FOR BIOMEDICAL RESEARCH 119 K. ARAI AND S. WATANABE SIGNAL TRANSDUCTION
MECHANISMS 10 MOLECULAR MECHANISMS OF REGULATORY SIGNAL TRANSDUCTION 133
E.S. SEVERIN AND M.V. NESTEROVA 11 MOLECULAR DIVERSITY OF SIGNAL
TRANSDUCTION SYSTEMS: A PUZZLE FOR PHARMACOLOGISTS OF TODAY AND TOMORROW
145 J. BOCKAERT PART 3: PHARMACOPHORE STUDIES PHARMACOPHORE MIMICKRY
MODELLING 12 THE FUTURE OF COMPUTER-AIDED DRUG DESIGN 163 G.R. MARSHALL
13 PHARMACOPHORE IDENTIFICATION BASED ON MOLECULAR ELECTROSTATIC
POTENTIALS (MEPS) 181 H.-D. HOLTJE 14 NEW RATIONAL APPROACHES FOR
STRUCTURE-ACTIVITY RELATIONSHIPS AND DRUG DESIGN 191 A. ITAI, N.
TOMIOKA, Y. KATO, Y. NISHIBATA AND S. SAITO SYNTHESIS OF PEPTIDOMIMETICS
15 RATIONAL DESIGN OF PEPTIDOMIMETICS: STRUCTURAL AND PHARMACOLOGICAL
ASPECTS 215 P.W. SCHILLER 16 NON-PEPTIDE LIGANDS FOR PEPTIDE RECEPTORS
233 R.M. FREIDINGER 17 PEPTIDOMIMETIC RESEARCH, DESIGN AND SYNTHESIS 247
W.F. HUFFMAN 18 PEPTIDOMIMETICS AS TOOLS FOR THE INITIATION AND ANALYSIS
OF PEPTIDE AND PROTEIN SECONDARY STRUCTURE: THE PROSPECTS FOR UNNATURAL
PROTEINS BY DESIGN 259 D.S. KEMP CONTENTS VII OPTIMIZATION 19 ON THE
FUTURE OF QSAR 281 C. HANSCH 20 COMPUTER-ASSISTED DRUG DESIGN IN THE
21ST CENTURY 295 Y.C. MARTIN, K.-H. KIM AND M.G. BURES PART 4:
BIOAVAILABILITY MANIPULATIONS PRODRUGS 2 1 TRENDS IN DESIGN OF PRODRUGS
FOR IMPROVED DRUG DELIVERY 321 H. BUNDGAARD DRUG TARGETING 22
ANTIBODY-BASED DRUG TARGETING APPROACHES: PERSPECTIVES AND CHALLENGES
351 D.J.A. CROMMELIN, J. BERGERS AND J. ZUIDEMA 23 NOVEL DRUG-DELIVERY
SYSTEMS 367 R. KIRSH AND G. WILSON 24 LIPID MICROSPHERE PREPARATIONS AND
LECITHINIZED PEPTIDES FOR DRUG-DELIVERY SYSTEMS 381 Y. MIZUSHIMA AND R.
IGARASHI INDEX 399
|
any_adam_object | 1 |
building | Verbundindex |
bvnumber | BV007922005 |
callnumber-first | R - Medicine |
callnumber-label | RS403 |
callnumber-raw | RS403 |
callnumber-search | RS403 |
callnumber-sort | RS 3403 |
callnumber-subject | RS - Pharmacy |
classification_rvk | VS 5000 |
ctrlnum | (OCoLC)25316862 (DE-599)BVBBV007922005 |
dewey-full | 615/.19 |
dewey-hundreds | 600 - Technology (Applied sciences) |
dewey-ones | 615 - Pharmacology and therapeutics |
dewey-raw | 615/.19 |
dewey-search | 615/.19 |
dewey-sort | 3615 219 |
dewey-tens | 610 - Medicine and health |
discipline | Chemie / Pharmazie Medizin |
edition | 1. publ. |
format | Book |
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isbn | 0632034084 |
language | English |
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physical | XII, 402 S. Ill., graph. Darst. |
publishDate | 1992 |
publishDateSearch | 1992 |
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publisher | Blackwell Scientific Publ. |
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series2 | A "Chemistry for the 21st century" monograph |
spelling | Medicinal chemistry for the 21st century International Union of Pure and Applied Chemistry. Ed. by C. G. Wermuth 1. publ. Oxford u.a. Blackwell Scientific Publ. 1992 XII, 402 S. Ill., graph. Darst. txt rdacontent n rdamedia nc rdacarrier A "Chemistry for the 21st century" monograph Chimie pharmaceutique Chimie pharmaceutique - Prévision Medische chemie gtt Quimica farmaceutica larpcal Chemistry, Pharmaceutical trends Pharmaceutical chemistry Pharmaceutical chemistry Forecasting Arzneimittelentwicklung (DE-588)4143176-5 gnd rswk-swf Arzneimitteldesign (DE-588)4278218-1 gnd rswk-swf Pharmazeutische Chemie (DE-588)4132158-3 gnd rswk-swf Forschungsplanung (DE-588)4155051-1 gnd rswk-swf Arzneimittel (DE-588)4003115-9 gnd rswk-swf Struktur-Aktivitäts-Beziehung (DE-588)4183784-8 gnd rswk-swf Bioverfügbarkeit (DE-588)4145660-9 gnd rswk-swf (DE-588)4143413-4 Aufsatzsammlung gnd-content Bioverfügbarkeit (DE-588)4145660-9 s DE-604 Struktur-Aktivitäts-Beziehung (DE-588)4183784-8 s Arzneimittel (DE-588)4003115-9 s Arzneimitteldesign (DE-588)4278218-1 s Arzneimittelentwicklung (DE-588)4143176-5 s Pharmazeutische Chemie (DE-588)4132158-3 s Forschungsplanung (DE-588)4155051-1 s Wermuth, Camille Georges Sonstige oth International Union of Pure and Applied Chemistry Sonstige (DE-588)1011135-9 oth GBV Datenaustausch application/pdf http://bvbr.bib-bvb.de:8991/F?func=service&doc_library=BVB01&local_base=BVB01&doc_number=005234945&sequence=000001&line_number=0001&func_code=DB_RECORDS&service_type=MEDIA Inhaltsverzeichnis |
spellingShingle | Medicinal chemistry for the 21st century Chimie pharmaceutique Chimie pharmaceutique - Prévision Medische chemie gtt Quimica farmaceutica larpcal Chemistry, Pharmaceutical trends Pharmaceutical chemistry Pharmaceutical chemistry Forecasting Arzneimittelentwicklung (DE-588)4143176-5 gnd Arzneimitteldesign (DE-588)4278218-1 gnd Pharmazeutische Chemie (DE-588)4132158-3 gnd Forschungsplanung (DE-588)4155051-1 gnd Arzneimittel (DE-588)4003115-9 gnd Struktur-Aktivitäts-Beziehung (DE-588)4183784-8 gnd Bioverfügbarkeit (DE-588)4145660-9 gnd |
subject_GND | (DE-588)4143176-5 (DE-588)4278218-1 (DE-588)4132158-3 (DE-588)4155051-1 (DE-588)4003115-9 (DE-588)4183784-8 (DE-588)4145660-9 (DE-588)4143413-4 |
title | Medicinal chemistry for the 21st century |
title_auth | Medicinal chemistry for the 21st century |
title_exact_search | Medicinal chemistry for the 21st century |
title_full | Medicinal chemistry for the 21st century International Union of Pure and Applied Chemistry. Ed. by C. G. Wermuth |
title_fullStr | Medicinal chemistry for the 21st century International Union of Pure and Applied Chemistry. Ed. by C. G. Wermuth |
title_full_unstemmed | Medicinal chemistry for the 21st century International Union of Pure and Applied Chemistry. Ed. by C. G. Wermuth |
title_short | Medicinal chemistry for the 21st century |
title_sort | medicinal chemistry for the 21st century |
topic | Chimie pharmaceutique Chimie pharmaceutique - Prévision Medische chemie gtt Quimica farmaceutica larpcal Chemistry, Pharmaceutical trends Pharmaceutical chemistry Pharmaceutical chemistry Forecasting Arzneimittelentwicklung (DE-588)4143176-5 gnd Arzneimitteldesign (DE-588)4278218-1 gnd Pharmazeutische Chemie (DE-588)4132158-3 gnd Forschungsplanung (DE-588)4155051-1 gnd Arzneimittel (DE-588)4003115-9 gnd Struktur-Aktivitäts-Beziehung (DE-588)4183784-8 gnd Bioverfügbarkeit (DE-588)4145660-9 gnd |
topic_facet | Chimie pharmaceutique Chimie pharmaceutique - Prévision Medische chemie Quimica farmaceutica Chemistry, Pharmaceutical trends Pharmaceutical chemistry Pharmaceutical chemistry Forecasting Arzneimittelentwicklung Arzneimitteldesign Pharmazeutische Chemie Forschungsplanung Arzneimittel Struktur-Aktivitäts-Beziehung Bioverfügbarkeit Aufsatzsammlung |
url | http://bvbr.bib-bvb.de:8991/F?func=service&doc_library=BVB01&local_base=BVB01&doc_number=005234945&sequence=000001&line_number=0001&func_code=DB_RECORDS&service_type=MEDIA |
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