Plasma binding of drugs and its consequences: proceedings of an International Symposium held on the occasion of the centenary of the Heymans Institute of Pharmacology, University of Ghent, Belgium, Ghent, September 27-28, 1990
Gespeichert in:
Format: | Buch |
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Sprache: | English |
Veröffentlicht: |
Ghent
Academia Press
1991
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Schlagworte: | |
Online-Zugang: | Inhaltsverzeichnis |
Beschreibung: | XXII, 259 S. graph. Darst. |
ISBN: | 9038200188 |
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adam_text | PLASMA BINDING OF DRUGS AND ITS CONSEQUENCES PROCEEDINGS OF AN
INTERNATIONAL SYMPOSIUM HELD ON THE OCCASION OF THE CENTENARY OF THE
HEYMANS INSTITUTE OF PHARMACOLOGY UNIVERSITY OF GHENT, BELGIUM GHENT,
SEPTEMBER 27-28, 1990 EDITORS: F. BELPAIRE, HEYMANS INSTITUTE OF
PHARMACOLOGY, UNIVERSITY OF GHENT, GHENT, BELGIUM M. BOGAERT, HEYMANS
INSTITUTE OF PHARMACOLOGY, UNIVERSITY OF GHENT, GHENT, BELGIUM J. P.
TILLEMENT, DEPARTEMENT DE PHARMACOLOGIE, UNIVERSITE DE PARIS XII,
CRETEIL, FRANCE R. VERBEECK, SCHOOL OF PHARMACY, CATHOLIC UNIVERSITY
OFLOUVAIN, BRUSSELS, BELGIUM 1991 ACADEMIA PRESS / GHENT CONTENTS
PREFACE V INTRODUCTION VII LIST OF PARTICIPANTS IX PART 1 TYPES AND
MECHANISMS OF DRUG BINDING THERMODYNAMIC ASPECTS OF DRUG-PROTEIN
INTERACTIONS: ACCEPTORS AND EFFECTORS 3 TESTA B. AND VAN GELDEREN J.G.
STOPPED-FLOW KINETIC ANALYSIS OF DRUG BINDING TO HUMAN SERUM ALBUMIN 11
RLETBROCK N., WORNER W. AND WOODCOCK B.G. BRAIN TISSUE EXTRACTION OF
PLASMA-BOUND DRUGS AND RATE CONSTANTS OF BINDING AND TRANSFER REACTIONS
21 URIENS. ANALYSIS OF OBSERVED BINDING EQUILIBRIUM DATA IN TERMS OF
SEVERAL ACCEPTABLE SETS OF BINDING CONSTANTS V 31 BRODERSEN R, VORUM H.
AND PEDERSEN A.O. TYPES OF B-ADRENERGIC BINDING SITES ON PLASMA PROTEINS
AND BLOOD CELLS 43 SAGER G. PART 2 VARIABILITY IN DRUG BINDING SPECIES
DIFFERENCES IN THE INDUCTION OF OC,-ACID GLYCOPROTEIN BY DRUGS 57
ABRAMSON F.P. PHARMACOGENETICS OF DRUG BINDING TO ALBUMIN AND EAP C.B.
AND BAUMANN P. XVII CONTENTS THE INFLUENCE OF SPECIES DIFFERENCES IN
DRUG-PROTEIN BINDING ON PHARMACOKINETIC SCALING 83 LIMA, J. J. DRUG
BINDING IN RENAL DISEASE 103 LINDUP W.E., HENDERSON S.J. AND BARKER C.E.
PLASMA PROTEIN BINDING OF DRUGS IN THE ELDERLY PATIENT 121 VERBEECK R.K.
PART 3 PHARMACOKINETIC, PHARMACODYNAMIC AND CLINICAL ASPECTS OF DRUG
BINDING STEREOSELECTIVITY OF PLASMA PROTEIN BINDING AND ITS
PHARMACOKINETIC CONSEQUENCES 137 BELPAIRE F.M., VERMEULEN A.M. AND
BOGAERT M.G. TISSUE BINDING OF DRUGS: METHODS OF DETERMINATION AND
PHARMACOKINETIC CONSEQUENCES 149 FICHTL B. DRUG BINDING AND
PHARMACOLOGIC ACTIVITY OF 01,-ADRENERGIC ANTAGONISTS 159 0M S . AND
CHIANG J PROTEIN BINDING OF ANTIBIOTICS AND ANTIMICROBIAL EFFICACY 171
MATTE H. THE ROLE OF PLASMA PROTEIN BINDING IN THE TRYPANOCIDAL ACTION
OF SURAMIN 179 WILTING J., COPPENS I., OPPERDOES F.R. AND VANSTERKENBURG
E.L.M. THE INFLUENCE OF PROTEIN BINDING ON VASOACTIVITY 191 ANDREASEN F.
AND CHRISTIANSEN E.H. THE CLINICAL CONSEQUENCES OF ALTERED PLASMA
PROTEIN BINDING 207 ROUTLEDGE P.A. CONCLUSIONS 219 TLIXEMENT J.P. PART 4
ABSTRACTS OF POSTERS BRAIN UPTAKE OF MIFEPRISTONE: EFFECT OF PROTEIN
BINDING 223 BELAIBA R, ZINI R, URIEN S AND TILLEMENT JP, XVNI CONTENTS
BINDING OF ALFENTANIL TO HUMAN OTJ-ACID GLYCOPROTEIN, ALBUMIN AND SERUM
224 BELPAIRE FM AND BOGAERT MG HSA BINDING OF 5 OXICAMS (NSDAID S) -
RELATIONSHIP WITH PHYSICOCHEMICAL PARAMETERS 225 BREE F, BECHALANY A,
NGUYEN P, TESTA B, TILLEMENT JP BINDING OF SR 33557 TO SERUM ALBUMINS: A
FLUORESCENCE STUDY 226 CHATELAIN P, LARUEL R AND MATTEAZZI JR,
CONFORMATION-LINKED STEROID BINDING PROPERTIES OF HUMAN SERUM ALBUMIN
227 FISCHER MJE, BOS OJM, WILTING J AND JANSSEN LHM INFLUENCE OF HUMAN
A,-ACID GLYCOPROTEIN BINDING AND SPECIFIC HUMAN TISSUE BINDING OF
MIFEPRISTONE ON ITS DISTRIBUTION IN HUMANS 228 GRIMALDI B AND TILLEMENT
JP BINDING OF A FURAN DICARBOXYLIC ACID TO HUMAN ALBUMIN - EFFECT OF
WARFARIN AND DANSYL SARCOSINE 229 HENDERSON SJ AND LINDUP WE, ROLE OF
PLASMA PROTEIN BINDING IN THE PHARMACOLOGICAL EVALUATION OF IN VIVO
MEASUREMENTS OF ANTICONVULSANT EFFECT INTENSITY 230 HOOGERKAMP A, ARENDS
RHGP, VOSKUYL RA AND DANHOF M A STUDY OF ISOPRENALINE BINDING TO A,-ACID
GLYCOPROTEIN BY THE FLUORESCENCE TECHNIQUE 231 JOHANSEN A-K, WLLLASSEN
N-P AND SAGER G , EFFECT OF CHRONIC DEXAMETHASONE TREATMENT ON
BLOOD-BRAIN BARRIER TRANSFER OF DRUGS 232 JOLLIET-RLANT P, CAULIN E,
BARR J, DAGHFOUS R AND TILLEMENT JP CEREBROSPINAL FLUID PHARMACOKINETICS
OF LUMBAR INTRATHECAL BACLOFERI; RELATIONSHIP WITH PHARMACODYNAMIC
PARAMETERS AND THERAPEUTIC EFFECTS IN MULTIPLE SCLEROSIS 233
JOLLIET-RIANT P, DECQ P, VILLAFANE R, SIOUFI A, LEPRESLE E, VERROUST J,
KERAVEL Y AND TILLEMENT JP TAMOXIFEN UPTAKE IN BRAIN TISSUE AND BRAIN
METASTASES 234 LIEN EA, WESTER K, LONNING PE, SOLHEIM E AND UELAND PM
PLASMA PROTEIN BINDING AND BLOOD DISTRIBUTION OF NEBIVOLOL IN RAT, DOG
AND HUMAN 235 MANNENS G, MEULDERMANS W, MOSTMANS E, VERBOVEN P AND
HEYKANTS J BINDING OF RETELLIPTINE, A NEW ANTITUMORAL AGENT, TO SERUM
PROTEINS AND ERYTHROCYTES 237 MAULARD C, BASTIAN G, URIEN SAND TILLEMENT
JP XIX CONTENTS SKIN AND PLASMA PROTEIN BINDING OF DRUGS ENHANCES
PERCUTANEOUS PENETRATION 238 MENCZELE, INTERACTION OF PIRPROFEN
ENANTIOMERS WITH HUMAN SERUM ALBUMIN 239 ORAVCOVA J, MLYNARK V,
BYSTRICKY S AND TRNOVEC T BINDING OF LAURATE TO HUMAN ALBUMIN 240
PEDERSEN AO, VORUM H AND BRODERSEN R DOES NON-ENZYMATIC GLYCOSYLATION
AFFECT DRUG BINDING PROPERTIES AT THE BENZODIAZEPINE BINDING SITE OF
HUMAN SERUM ALBUMIN? 241 PFLEIDERER S, WORNER W AND RIETBROCK N PROTEIN
BINDING OF METHOTREXATE ON HUMAN ALBUMIN AND SERUM: A FIRST DERIVATIVE
SPECTROSCOPIC ANALYSIS 242 ROCHAS MA, TUFENKJI AE, LEVILLAIN P AND HOUIN
G QUALITATIVE CHANGES OF AAG AND THEIR INFLUENCE ON SERUM PROTEIN DRUG
BINDING 243 RODRFGUEZ-SASIAFN JM, AGUIRRE C AND CALVO R DOES BINDING OF
DRUG TO MILK PROTEINS DETERMINE THE EXTENT OF DRUG EXCRETION INTO MILK?
244 STEBLER T AND GUENTERT TW, DIFFERENCES IN LIGAND DISPLACEMENT FOR
DIFFERENT METHODS USED IN THE DEPROTEINIZATION OF UREMIC SERA 245
VANHOLDER R, HOFLIGER N, DE SMET R AND RINGOIR S FACTORS AFFECTING
PROTEIN BINDING OF THEOPHYLLINE AND PHENYTOIN IN CHRONIC RENAL FAILURE
246 VANHOLDER R, VAN LANDSCHOOT N, DE SMET R, HOFLIGER N AND RINGOIR S
THE EFFECT OF AGE ON THE SERUM CONCENTRATION OF ALBUMIN AND (
GLYCOPROTEIN 247 VEERING BTH, BURM AGL, SOUVERIJN JHM AND SPIERDIJK J
THE EFFECT OF AGING ON PLASMA PROTEIN BINDING AND TISSUE DISTRIBUTION OF
R- AND S-PROPRANOLOL IN THE RAT 248 VERMEULEN A, BELPAIRE F, DE SMET F,
MOERMAN E AND BOGAERT M BINDING OF DIAZEPAM, SALICYLIC ACID AND
DIGITOXIN TO ALBUMIN ISOLATED FROM UMBILICAL CORD AND ADULT PLASMA 249
VIANI A, CAPPELLO M, SILVESTRI D AND PACIFICI GM, DIFFERENTIAL EFFECT OF
AGING ON ALBUMIN CONCENTRATION AND PROTEIN BINDING OF DIAZEPAM AND
SALICYLIC ACID IN HEALTHY SUBJECTS AND RENAL PATIENTS 250 VIANI A, RIZZO
G, CARRAI M AND PACIFICI GM, XX CONTENTS HIGH- AND LOW-AFFINITY HUMAN
ALBUMIN IN A COMMERCIAL PREPARATION 251 VORUM H, PEDERSEN AO AND
BRODERSEN R THE REDUCTION IN PROTEIN BINDING OF HIGHLY BOUND
SULFONAMIDES BY NJ-GLUCURONIDATION IN MAN 252 VREE TB, BENEKEN KOLMER
EWJ, MARTEA M AND BAARS AM STOPPED-FLOW STUDIES ON THE KINETICS OF DRUG
BINDING TO HUMAN SERUM ALBUMIN 253 WORNER W, PFLEIDERER S AND RLETBROCK
N REAPPRAISAL OF SALICYLATE BINDING TO HUMAN SERUM ALBUMIN: IMIDAZOLE
SALICYLATE AS AN EXAMPLE 254 ZINI R, MORIN D, ACUTO GC, BIANCHINI C AND
TILLEMENT JP INDEX 255 XXI
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spelling | Plasma binding of drugs and its consequences proceedings of an International Symposium held on the occasion of the centenary of the Heymans Institute of Pharmacology, University of Ghent, Belgium, Ghent, September 27-28, 1990 eds.: F. Belpaire ... Ghent Academia Press 1991 XXII, 259 S. graph. Darst. txt rdacontent n rdamedia nc rdacarrier Bloedplasma gtt Geneesmiddelen gtt Blood Proteins metabolism Congresses Drugs Absorption and adsorption Congresses Drugs Metabolism Congresses Pharmaceutical Preparations metabolism Congresses Protein Binding physiology Congresses Protein binding Congresses Plasmaproteine (DE-588)4127411-8 gnd rswk-swf Arzneistoffträger (DE-588)4278196-6 gnd rswk-swf (DE-588)1071861417 Konferenzschrift 1990 Genf gnd-content Plasmaproteine (DE-588)4127411-8 s Arzneistoffträger (DE-588)4278196-6 s DE-604 Belpaire, F. M. Sonstige oth GBV Datenaustausch application/pdf http://bvbr.bib-bvb.de:8991/F?func=service&doc_library=BVB01&local_base=BVB01&doc_number=005062347&sequence=000001&line_number=0001&func_code=DB_RECORDS&service_type=MEDIA Inhaltsverzeichnis |
spellingShingle | Plasma binding of drugs and its consequences proceedings of an International Symposium held on the occasion of the centenary of the Heymans Institute of Pharmacology, University of Ghent, Belgium, Ghent, September 27-28, 1990 Bloedplasma gtt Geneesmiddelen gtt Blood Proteins metabolism Congresses Drugs Absorption and adsorption Congresses Drugs Metabolism Congresses Pharmaceutical Preparations metabolism Congresses Protein Binding physiology Congresses Protein binding Congresses Plasmaproteine (DE-588)4127411-8 gnd Arzneistoffträger (DE-588)4278196-6 gnd |
subject_GND | (DE-588)4127411-8 (DE-588)4278196-6 (DE-588)1071861417 |
title | Plasma binding of drugs and its consequences proceedings of an International Symposium held on the occasion of the centenary of the Heymans Institute of Pharmacology, University of Ghent, Belgium, Ghent, September 27-28, 1990 |
title_auth | Plasma binding of drugs and its consequences proceedings of an International Symposium held on the occasion of the centenary of the Heymans Institute of Pharmacology, University of Ghent, Belgium, Ghent, September 27-28, 1990 |
title_exact_search | Plasma binding of drugs and its consequences proceedings of an International Symposium held on the occasion of the centenary of the Heymans Institute of Pharmacology, University of Ghent, Belgium, Ghent, September 27-28, 1990 |
title_full | Plasma binding of drugs and its consequences proceedings of an International Symposium held on the occasion of the centenary of the Heymans Institute of Pharmacology, University of Ghent, Belgium, Ghent, September 27-28, 1990 eds.: F. Belpaire ... |
title_fullStr | Plasma binding of drugs and its consequences proceedings of an International Symposium held on the occasion of the centenary of the Heymans Institute of Pharmacology, University of Ghent, Belgium, Ghent, September 27-28, 1990 eds.: F. Belpaire ... |
title_full_unstemmed | Plasma binding of drugs and its consequences proceedings of an International Symposium held on the occasion of the centenary of the Heymans Institute of Pharmacology, University of Ghent, Belgium, Ghent, September 27-28, 1990 eds.: F. Belpaire ... |
title_short | Plasma binding of drugs and its consequences |
title_sort | plasma binding of drugs and its consequences proceedings of an international symposium held on the occasion of the centenary of the heymans institute of pharmacology university of ghent belgium ghent september 27 28 1990 |
title_sub | proceedings of an International Symposium held on the occasion of the centenary of the Heymans Institute of Pharmacology, University of Ghent, Belgium, Ghent, September 27-28, 1990 |
topic | Bloedplasma gtt Geneesmiddelen gtt Blood Proteins metabolism Congresses Drugs Absorption and adsorption Congresses Drugs Metabolism Congresses Pharmaceutical Preparations metabolism Congresses Protein Binding physiology Congresses Protein binding Congresses Plasmaproteine (DE-588)4127411-8 gnd Arzneistoffträger (DE-588)4278196-6 gnd |
topic_facet | Bloedplasma Geneesmiddelen Blood Proteins metabolism Congresses Drugs Absorption and adsorption Congresses Drugs Metabolism Congresses Pharmaceutical Preparations metabolism Congresses Protein Binding physiology Congresses Protein binding Congresses Plasmaproteine Arzneistoffträger Konferenzschrift 1990 Genf |
url | http://bvbr.bib-bvb.de:8991/F?func=service&doc_library=BVB01&local_base=BVB01&doc_number=005062347&sequence=000001&line_number=0001&func_code=DB_RECORDS&service_type=MEDIA |
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