Affinity and efficacy: the components of drug-receptor interactions = Components of drug-receptor interactions
Gespeichert in:
1. Verfasser: | |
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Format: | Elektronisch E-Book |
Sprache: | English |
Veröffentlicht: |
New Jersey
World Scientific
[2014]
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Schlagworte: | |
Online-Zugang: | FAW01 FAW02 |
Beschreibung: | Print version record |
Beschreibung: | 1 online resource |
ISBN: | 9789814324229 9814324221 9789814322560 9814322563 |
Internformat
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245 | 1 | 0 | |a Affinity and efficacy |b the components of drug-receptor interactions = Components of drug-receptor interactions |c Frederick J. Ehlert |
246 | 1 | 3 | |a Components of drug-receptor interactions |
246 | 1 | 1 | |a Components of drug-receptor interactions |
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505 | 8 | |a Ligand-gated ion channels -- Affinity and efficacy of orthosteric ligands at ligand-gated ion channels -- Competitive interactions between orthostheric ligands at ligand-gated ion channels -- Analysis of allosteric interactions at ligand-gated ion channels -- G protein-coupled receptors and G protein signaling -- Affinity and efficacy of the agonist-receptor-G-protein interaction -- Estimating affinity and efficacy by reverse-engineering and response-clamp analysis -- Analysis of agonism and inverse agonism in signaling pathways that exhibit constitutive activity -- Analysis of ligand bias in receptor signaling through different G protein pathways -- Competitive interactions between orthosteric ligands in functional assays on G protein-coupled receptors -- Analysis of allosterism in functional assays on G protein-coupled receptors -- Analysis of drug-receptor interactions using radioligand binding assays on G protein-coupled receptors | |
650 | 4 | |a Receptors, Drug | |
650 | 4 | |a Ligand-Gated Ion Channels | |
650 | 4 | |a Protein Binding | |
650 | 4 | |a Radioligand Assay | |
650 | 4 | |a Receptors, G-Protein-Coupled | |
650 | 7 | |a MEDICAL / Pharmacology |2 bisacsh | |
650 | 7 | |a Drug-nutrient interactions |2 fast | |
650 | 7 | |a Drug receptors |2 fast | |
650 | 7 | |a Drugs / Effectiveness |2 fast | |
650 | 7 | |a Pharmaceutical chemistry |2 fast | |
650 | 4 | |a Drug receptors | |
650 | 4 | |a Medizin | |
650 | 4 | |a Drug receptors |a Drugs |x Effectiveness |a Drug-nutrient interactions |a Pharmaceutical chemistry | |
776 | 0 | 8 | |i Erscheint auch als |n Druck-Ausgabe |a Ehlert, Frederick J |t . Affinity and efficacy |
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Datensatz im Suchindex
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any_adam_object | |
author | Ehlert, Frederick J. |
author_facet | Ehlert, Frederick J. |
author_role | aut |
author_sort | Ehlert, Frederick J. |
author_variant | f j e fj fje |
building | Verbundindex |
bvnumber | BV043783693 |
collection | ZDB-4-EBA |
contents | Ligand-gated ion channels -- Affinity and efficacy of orthosteric ligands at ligand-gated ion channels -- Competitive interactions between orthostheric ligands at ligand-gated ion channels -- Analysis of allosteric interactions at ligand-gated ion channels -- G protein-coupled receptors and G protein signaling -- Affinity and efficacy of the agonist-receptor-G-protein interaction -- Estimating affinity and efficacy by reverse-engineering and response-clamp analysis -- Analysis of agonism and inverse agonism in signaling pathways that exhibit constitutive activity -- Analysis of ligand bias in receptor signaling through different G protein pathways -- Competitive interactions between orthosteric ligands in functional assays on G protein-coupled receptors -- Analysis of allosterism in functional assays on G protein-coupled receptors -- Analysis of drug-receptor interactions using radioligand binding assays on G protein-coupled receptors |
ctrlnum | (ZDB-4-EBA)ocn898070271 (OCoLC)898070271 (DE-599)BVBBV043783693 |
dewey-full | 615.7/0452 |
dewey-hundreds | 600 - Technology (Applied sciences) |
dewey-ones | 615 - Pharmacology and therapeutics |
dewey-raw | 615.7/0452 |
dewey-search | 615.7/0452 |
dewey-sort | 3615.7 3452 |
dewey-tens | 610 - Medicine and health |
discipline | Medizin |
format | Electronic eBook |
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id | DE-604.BV043783693 |
illustrated | Not Illustrated |
indexdate | 2024-07-10T07:35:00Z |
institution | BVB |
isbn | 9789814324229 9814324221 9789814322560 9814322563 |
language | English |
oai_aleph_id | oai:aleph.bib-bvb.de:BVB01-029194753 |
oclc_num | 898070271 |
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owner_facet | DE-1046 DE-1047 |
physical | 1 online resource |
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publishDate | 2014 |
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publisher | World Scientific |
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spelling | Ehlert, Frederick J. Verfasser aut Affinity and efficacy the components of drug-receptor interactions = Components of drug-receptor interactions Frederick J. Ehlert Components of drug-receptor interactions New Jersey World Scientific [2014] 1 online resource txt rdacontent c rdamedia cr rdacarrier Print version record Ligand-gated ion channels -- Affinity and efficacy of orthosteric ligands at ligand-gated ion channels -- Competitive interactions between orthostheric ligands at ligand-gated ion channels -- Analysis of allosteric interactions at ligand-gated ion channels -- G protein-coupled receptors and G protein signaling -- Affinity and efficacy of the agonist-receptor-G-protein interaction -- Estimating affinity and efficacy by reverse-engineering and response-clamp analysis -- Analysis of agonism and inverse agonism in signaling pathways that exhibit constitutive activity -- Analysis of ligand bias in receptor signaling through different G protein pathways -- Competitive interactions between orthosteric ligands in functional assays on G protein-coupled receptors -- Analysis of allosterism in functional assays on G protein-coupled receptors -- Analysis of drug-receptor interactions using radioligand binding assays on G protein-coupled receptors Receptors, Drug Ligand-Gated Ion Channels Protein Binding Radioligand Assay Receptors, G-Protein-Coupled MEDICAL / Pharmacology bisacsh Drug-nutrient interactions fast Drug receptors fast Drugs / Effectiveness fast Pharmaceutical chemistry fast Drug receptors Medizin Drug receptors Drugs Effectiveness Drug-nutrient interactions Pharmaceutical chemistry Erscheint auch als Druck-Ausgabe Ehlert, Frederick J . Affinity and efficacy |
spellingShingle | Ehlert, Frederick J. Affinity and efficacy the components of drug-receptor interactions = Components of drug-receptor interactions Ligand-gated ion channels -- Affinity and efficacy of orthosteric ligands at ligand-gated ion channels -- Competitive interactions between orthostheric ligands at ligand-gated ion channels -- Analysis of allosteric interactions at ligand-gated ion channels -- G protein-coupled receptors and G protein signaling -- Affinity and efficacy of the agonist-receptor-G-protein interaction -- Estimating affinity and efficacy by reverse-engineering and response-clamp analysis -- Analysis of agonism and inverse agonism in signaling pathways that exhibit constitutive activity -- Analysis of ligand bias in receptor signaling through different G protein pathways -- Competitive interactions between orthosteric ligands in functional assays on G protein-coupled receptors -- Analysis of allosterism in functional assays on G protein-coupled receptors -- Analysis of drug-receptor interactions using radioligand binding assays on G protein-coupled receptors Receptors, Drug Ligand-Gated Ion Channels Protein Binding Radioligand Assay Receptors, G-Protein-Coupled MEDICAL / Pharmacology bisacsh Drug-nutrient interactions fast Drug receptors fast Drugs / Effectiveness fast Pharmaceutical chemistry fast Drug receptors Medizin Drug receptors Drugs Effectiveness Drug-nutrient interactions Pharmaceutical chemistry |
title | Affinity and efficacy the components of drug-receptor interactions = Components of drug-receptor interactions |
title_alt | Components of drug-receptor interactions |
title_auth | Affinity and efficacy the components of drug-receptor interactions = Components of drug-receptor interactions |
title_exact_search | Affinity and efficacy the components of drug-receptor interactions = Components of drug-receptor interactions |
title_full | Affinity and efficacy the components of drug-receptor interactions = Components of drug-receptor interactions Frederick J. Ehlert |
title_fullStr | Affinity and efficacy the components of drug-receptor interactions = Components of drug-receptor interactions Frederick J. Ehlert |
title_full_unstemmed | Affinity and efficacy the components of drug-receptor interactions = Components of drug-receptor interactions Frederick J. Ehlert |
title_short | Affinity and efficacy |
title_sort | affinity and efficacy the components of drug receptor interactions components of drug receptor interactions |
title_sub | the components of drug-receptor interactions = Components of drug-receptor interactions |
topic | Receptors, Drug Ligand-Gated Ion Channels Protein Binding Radioligand Assay Receptors, G-Protein-Coupled MEDICAL / Pharmacology bisacsh Drug-nutrient interactions fast Drug receptors fast Drugs / Effectiveness fast Pharmaceutical chemistry fast Drug receptors Medizin Drug receptors Drugs Effectiveness Drug-nutrient interactions Pharmaceutical chemistry |
topic_facet | Receptors, Drug Ligand-Gated Ion Channels Protein Binding Radioligand Assay Receptors, G-Protein-Coupled MEDICAL / Pharmacology Drug-nutrient interactions Drug receptors Drugs / Effectiveness Pharmaceutical chemistry Medizin Drug receptors Drugs Effectiveness Drug-nutrient interactions Pharmaceutical chemistry |
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