High-throughput lead optimization in drug discovery:
Gespeichert in:
Format: | Buch |
---|---|
Sprache: | English |
Veröffentlicht: |
Boca Raton, Fla. [u.a.]
CRC Press
2008
|
Schriftenreihe: | Critical reviews in combinatorial chemistry
|
Schlagworte: | |
Online-Zugang: | Publisher description kostenfrei Inhaltsverzeichnis Inhaltsverzeichnis |
Beschreibung: | Literaturangaben |
Beschreibung: | IX, 243 S. Ill., graph. Darst. |
ISBN: | 9780849372681 |
Internformat
MARC
LEADER | 00000nam a2200000 c 4500 | ||
---|---|---|---|
001 | BV035541145 | ||
003 | DE-604 | ||
005 | 00000000000000.0 | ||
007 | t | ||
008 | 090528s2008 ad|| |||| 00||| eng d | ||
010 | |a 2007035804 | ||
020 | |a 9780849372681 |c hardback : alk. paper |9 978-0-8493-7268-1 | ||
035 | |a (OCoLC)166454429 | ||
035 | |a (DE-599)GBV543566048 | ||
040 | |a DE-604 |b ger | ||
041 | 0 | |a eng | |
049 | |a DE-19 | ||
050 | 0 | |a RS419.5 | |
082 | 0 | |a 615/.19 |2 22 | |
084 | |a VS 5350 |0 (DE-625)147687:253 |2 rvk | ||
245 | 1 | 0 | |a High-throughput lead optimization in drug discovery |c ed. by Tushar Kshirsagar |
264 | 1 | |a Boca Raton, Fla. [u.a.] |b CRC Press |c 2008 | |
300 | |a IX, 243 S. |b Ill., graph. Darst. | ||
336 | |b txt |2 rdacontent | ||
337 | |b n |2 rdamedia | ||
338 | |b nc |2 rdacarrier | ||
490 | 0 | |a Critical reviews in combinatorial chemistry | |
500 | |a Literaturangaben | ||
650 | 0 | |a High throughput screening (Drug development) | |
650 | 0 | |a Combinatorial chemistry | |
650 | 0 | |a Drug development | |
650 | 4 | |a Combinatorial Chemistry Techniques | |
650 | 4 | |a Combinatorial chemistry | |
650 | 4 | |a Databases, Genetic | |
650 | 4 | |a Drug Design | |
650 | 4 | |a Drug development | |
650 | 4 | |a Gene Library | |
650 | 4 | |a High throughput screening (Drug development) | |
650 | 0 | 7 | |a High throughput screening |0 (DE-588)4596131-1 |2 gnd |9 rswk-swf |
650 | 0 | 7 | |a Arzneimittelforschung |0 (DE-588)4003120-2 |2 gnd |9 rswk-swf |
650 | 0 | 7 | |a Kombinatorische Synthese |0 (DE-588)4513555-1 |2 gnd |9 rswk-swf |
689 | 0 | 0 | |a High throughput screening |0 (DE-588)4596131-1 |D s |
689 | 0 | 1 | |a Kombinatorische Synthese |0 (DE-588)4513555-1 |D s |
689 | 0 | 2 | |a Arzneimittelforschung |0 (DE-588)4003120-2 |D s |
689 | 0 | |5 DE-604 | |
700 | 1 | |a Kshirsagar, Tushar |e Sonstige |4 oth | |
856 | 4 | |u http://www.loc.gov/catdir/enhancements/fy0829/2007035804-d.html |y Publisher description |z kostenfrei | |
856 | 4 | |u http://www.loc.gov/catdir/toc/fy0804/2007035804.html |z kostenfrei |3 Inhaltsverzeichnis | |
856 | 4 | |m DE-601 |q pdf/application |u http://www.gbv.de/dms/bowker/toc/9780849372681.pdf |3 Inhaltsverzeichnis | |
856 | 4 | 2 | |m GBV Datenaustausch |q application/pdf |u http://bvbr.bib-bvb.de:8991/F?func=service&doc_library=BVB01&local_base=BVB01&doc_number=017597195&sequence=000001&line_number=0001&func_code=DB_RECORDS&service_type=MEDIA |3 Inhaltsverzeichnis |
999 | |a oai:aleph.bib-bvb.de:BVB01-017597195 |
Datensatz im Suchindex
_version_ | 1804139181188841472 |
---|---|
adam_text | IMAGE 1
INTRODUCTION AND REVIEW
P. 1
APPLICATION OF PARALLEL SYNTHESIS TO THE OPTIMIZATION OF INHIBITORS OF
THE ZIPA-FTSZ PROTEIN-PROTEIN INTERACTION
P. 85
CASE STUDIES OF PARALLEL SYNTHESIS IN HIT IDENTIFICATION, HIT
EXPLORATION, HIT-TO-LEAD, AND LEAD OPTIMIZATION PROGRAMS
P. 99
A SUCCESSFUL APPLICATION OF PARALLEL SYNTHESIS TO COMPUTER-ASSISTED
STRUCTURAL OPTIMIZATION OF NEW LEADS TARGETING HUMAN IMMUNODEFICIENCY
VIRUS-I REVERSE TRANSCRIPTASE: THE CASE OF ACYLTHIOCARBAMATES AND
THIOCARBAMATES
P. 117
HOW HIGH-THROUGHPUT MEDICINAL CHEMISTRY CAN EXPEDITE LEAD DISCOVERY,
LEAD OPTIMIZATION, AND BEYOND
P. 151
RAPID LEAD IDENTIFICATION OF INHIBITORS OF ADENINE NUCLEOTIDE
TRANSLOCASE: A CASE STUDY OF APPLYING COMBINATORIAL CHEMISTRY TECHNIQUES
IN DRUG DISCOVERY
P. 165
PARALLEL SYNTHESIS OF ANTICANCER, ANTIINFLAMMATORY, AND ANTIVIRAL AGENTS
DERIVED FROM L- AND D-AMINO ACIDS
P. 177
APPLICATION OF SOLID-PHASE PARALLEL SYNTHESIS IN LEAD OPTIMIZATION
STUDIES P. 195
HIGH-THROUGHPUT SOLID-PHASE SYNTHESIS OF NUCLEOSIDE-BASED LIBRARIES IN
THE SEARCH FOR NEW ANTIBIOTICS
P. 215
INDEX
P. 239
TABLE OF CONTENTS PROVIDED BY BLACKWELL S BOOK SERVICES AND R.R. BOWKER.
USED WITH PERMISSION.
|
any_adam_object | 1 |
building | Verbundindex |
bvnumber | BV035541145 |
callnumber-first | R - Medicine |
callnumber-label | RS419 |
callnumber-raw | RS419.5 |
callnumber-search | RS419.5 |
callnumber-sort | RS 3419.5 |
callnumber-subject | RS - Pharmacy |
classification_rvk | VS 5350 |
ctrlnum | (OCoLC)166454429 (DE-599)GBV543566048 |
dewey-full | 615/.19 |
dewey-hundreds | 600 - Technology (Applied sciences) |
dewey-ones | 615 - Pharmacology and therapeutics |
dewey-raw | 615/.19 |
dewey-search | 615/.19 |
dewey-sort | 3615 219 |
dewey-tens | 610 - Medicine and health |
discipline | Chemie / Pharmazie Medizin |
format | Book |
fullrecord | <?xml version="1.0" encoding="UTF-8"?><collection xmlns="http://www.loc.gov/MARC21/slim"><record><leader>02408nam a2200577 c 4500</leader><controlfield tag="001">BV035541145</controlfield><controlfield tag="003">DE-604</controlfield><controlfield tag="005">00000000000000.0</controlfield><controlfield tag="007">t</controlfield><controlfield tag="008">090528s2008 ad|| |||| 00||| eng d</controlfield><datafield tag="010" ind1=" " ind2=" "><subfield code="a">2007035804</subfield></datafield><datafield tag="020" ind1=" " ind2=" "><subfield code="a">9780849372681</subfield><subfield code="c">hardback : alk. paper</subfield><subfield code="9">978-0-8493-7268-1</subfield></datafield><datafield tag="035" ind1=" " ind2=" "><subfield code="a">(OCoLC)166454429</subfield></datafield><datafield tag="035" ind1=" " ind2=" "><subfield code="a">(DE-599)GBV543566048</subfield></datafield><datafield tag="040" ind1=" " ind2=" "><subfield code="a">DE-604</subfield><subfield code="b">ger</subfield></datafield><datafield tag="041" ind1="0" ind2=" "><subfield code="a">eng</subfield></datafield><datafield tag="049" ind1=" " ind2=" "><subfield code="a">DE-19</subfield></datafield><datafield tag="050" ind1=" " ind2="0"><subfield code="a">RS419.5</subfield></datafield><datafield tag="082" ind1="0" ind2=" "><subfield code="a">615/.19</subfield><subfield code="2">22</subfield></datafield><datafield tag="084" ind1=" " ind2=" "><subfield code="a">VS 5350</subfield><subfield code="0">(DE-625)147687:253</subfield><subfield code="2">rvk</subfield></datafield><datafield tag="245" ind1="1" ind2="0"><subfield code="a">High-throughput lead optimization in drug discovery</subfield><subfield code="c">ed. by Tushar Kshirsagar</subfield></datafield><datafield tag="264" ind1=" " ind2="1"><subfield code="a">Boca Raton, Fla. [u.a.]</subfield><subfield code="b">CRC Press</subfield><subfield code="c">2008</subfield></datafield><datafield tag="300" ind1=" " ind2=" "><subfield code="a">IX, 243 S.</subfield><subfield code="b">Ill., graph. Darst.</subfield></datafield><datafield tag="336" ind1=" " ind2=" "><subfield code="b">txt</subfield><subfield code="2">rdacontent</subfield></datafield><datafield tag="337" ind1=" " ind2=" "><subfield code="b">n</subfield><subfield code="2">rdamedia</subfield></datafield><datafield tag="338" ind1=" " ind2=" "><subfield code="b">nc</subfield><subfield code="2">rdacarrier</subfield></datafield><datafield tag="490" ind1="0" ind2=" "><subfield code="a">Critical reviews in combinatorial chemistry</subfield></datafield><datafield tag="500" ind1=" " ind2=" "><subfield code="a">Literaturangaben</subfield></datafield><datafield tag="650" ind1=" " ind2="0"><subfield code="a">High throughput screening (Drug development)</subfield></datafield><datafield tag="650" ind1=" " ind2="0"><subfield code="a">Combinatorial chemistry</subfield></datafield><datafield tag="650" ind1=" " ind2="0"><subfield code="a">Drug development</subfield></datafield><datafield tag="650" ind1=" " ind2="4"><subfield code="a">Combinatorial Chemistry Techniques</subfield></datafield><datafield tag="650" ind1=" " ind2="4"><subfield code="a">Combinatorial chemistry</subfield></datafield><datafield tag="650" ind1=" " ind2="4"><subfield code="a">Databases, Genetic</subfield></datafield><datafield tag="650" ind1=" " ind2="4"><subfield code="a">Drug Design</subfield></datafield><datafield tag="650" ind1=" " ind2="4"><subfield code="a">Drug development</subfield></datafield><datafield tag="650" ind1=" " ind2="4"><subfield code="a">Gene Library</subfield></datafield><datafield tag="650" ind1=" " ind2="4"><subfield code="a">High throughput screening (Drug development)</subfield></datafield><datafield tag="650" ind1="0" ind2="7"><subfield code="a">High throughput screening</subfield><subfield code="0">(DE-588)4596131-1</subfield><subfield code="2">gnd</subfield><subfield code="9">rswk-swf</subfield></datafield><datafield tag="650" ind1="0" ind2="7"><subfield code="a">Arzneimittelforschung</subfield><subfield code="0">(DE-588)4003120-2</subfield><subfield code="2">gnd</subfield><subfield code="9">rswk-swf</subfield></datafield><datafield tag="650" ind1="0" ind2="7"><subfield code="a">Kombinatorische Synthese</subfield><subfield code="0">(DE-588)4513555-1</subfield><subfield code="2">gnd</subfield><subfield code="9">rswk-swf</subfield></datafield><datafield tag="689" ind1="0" ind2="0"><subfield code="a">High throughput screening</subfield><subfield code="0">(DE-588)4596131-1</subfield><subfield code="D">s</subfield></datafield><datafield tag="689" ind1="0" ind2="1"><subfield code="a">Kombinatorische Synthese</subfield><subfield code="0">(DE-588)4513555-1</subfield><subfield code="D">s</subfield></datafield><datafield tag="689" ind1="0" ind2="2"><subfield code="a">Arzneimittelforschung</subfield><subfield code="0">(DE-588)4003120-2</subfield><subfield code="D">s</subfield></datafield><datafield tag="689" ind1="0" ind2=" "><subfield code="5">DE-604</subfield></datafield><datafield tag="700" ind1="1" ind2=" "><subfield code="a">Kshirsagar, Tushar</subfield><subfield code="e">Sonstige</subfield><subfield code="4">oth</subfield></datafield><datafield tag="856" ind1="4" ind2=" "><subfield code="u">http://www.loc.gov/catdir/enhancements/fy0829/2007035804-d.html</subfield><subfield code="y">Publisher description</subfield><subfield code="z">kostenfrei</subfield></datafield><datafield tag="856" ind1="4" ind2=" "><subfield code="u">http://www.loc.gov/catdir/toc/fy0804/2007035804.html</subfield><subfield code="z">kostenfrei</subfield><subfield code="3">Inhaltsverzeichnis</subfield></datafield><datafield tag="856" ind1="4" ind2=" "><subfield code="m">DE-601</subfield><subfield code="q">pdf/application</subfield><subfield code="u">http://www.gbv.de/dms/bowker/toc/9780849372681.pdf</subfield><subfield code="3">Inhaltsverzeichnis</subfield></datafield><datafield tag="856" ind1="4" ind2="2"><subfield code="m">GBV Datenaustausch</subfield><subfield code="q">application/pdf</subfield><subfield code="u">http://bvbr.bib-bvb.de:8991/F?func=service&doc_library=BVB01&local_base=BVB01&doc_number=017597195&sequence=000001&line_number=0001&func_code=DB_RECORDS&service_type=MEDIA</subfield><subfield code="3">Inhaltsverzeichnis</subfield></datafield><datafield tag="999" ind1=" " ind2=" "><subfield code="a">oai:aleph.bib-bvb.de:BVB01-017597195</subfield></datafield></record></collection> |
id | DE-604.BV035541145 |
illustrated | Illustrated |
indexdate | 2024-07-09T21:40:00Z |
institution | BVB |
isbn | 9780849372681 |
language | English |
lccn | 2007035804 |
oai_aleph_id | oai:aleph.bib-bvb.de:BVB01-017597195 |
oclc_num | 166454429 |
open_access_boolean | 1 |
owner | DE-19 DE-BY-UBM |
owner_facet | DE-19 DE-BY-UBM |
physical | IX, 243 S. Ill., graph. Darst. |
publishDate | 2008 |
publishDateSearch | 2008 |
publishDateSort | 2008 |
publisher | CRC Press |
record_format | marc |
series2 | Critical reviews in combinatorial chemistry |
spelling | High-throughput lead optimization in drug discovery ed. by Tushar Kshirsagar Boca Raton, Fla. [u.a.] CRC Press 2008 IX, 243 S. Ill., graph. Darst. txt rdacontent n rdamedia nc rdacarrier Critical reviews in combinatorial chemistry Literaturangaben High throughput screening (Drug development) Combinatorial chemistry Drug development Combinatorial Chemistry Techniques Databases, Genetic Drug Design Gene Library High throughput screening (DE-588)4596131-1 gnd rswk-swf Arzneimittelforschung (DE-588)4003120-2 gnd rswk-swf Kombinatorische Synthese (DE-588)4513555-1 gnd rswk-swf High throughput screening (DE-588)4596131-1 s Kombinatorische Synthese (DE-588)4513555-1 s Arzneimittelforschung (DE-588)4003120-2 s DE-604 Kshirsagar, Tushar Sonstige oth http://www.loc.gov/catdir/enhancements/fy0829/2007035804-d.html Publisher description kostenfrei http://www.loc.gov/catdir/toc/fy0804/2007035804.html kostenfrei Inhaltsverzeichnis DE-601 pdf/application http://www.gbv.de/dms/bowker/toc/9780849372681.pdf Inhaltsverzeichnis GBV Datenaustausch application/pdf http://bvbr.bib-bvb.de:8991/F?func=service&doc_library=BVB01&local_base=BVB01&doc_number=017597195&sequence=000001&line_number=0001&func_code=DB_RECORDS&service_type=MEDIA Inhaltsverzeichnis |
spellingShingle | High-throughput lead optimization in drug discovery High throughput screening (Drug development) Combinatorial chemistry Drug development Combinatorial Chemistry Techniques Databases, Genetic Drug Design Gene Library High throughput screening (DE-588)4596131-1 gnd Arzneimittelforschung (DE-588)4003120-2 gnd Kombinatorische Synthese (DE-588)4513555-1 gnd |
subject_GND | (DE-588)4596131-1 (DE-588)4003120-2 (DE-588)4513555-1 |
title | High-throughput lead optimization in drug discovery |
title_auth | High-throughput lead optimization in drug discovery |
title_exact_search | High-throughput lead optimization in drug discovery |
title_full | High-throughput lead optimization in drug discovery ed. by Tushar Kshirsagar |
title_fullStr | High-throughput lead optimization in drug discovery ed. by Tushar Kshirsagar |
title_full_unstemmed | High-throughput lead optimization in drug discovery ed. by Tushar Kshirsagar |
title_short | High-throughput lead optimization in drug discovery |
title_sort | high throughput lead optimization in drug discovery |
topic | High throughput screening (Drug development) Combinatorial chemistry Drug development Combinatorial Chemistry Techniques Databases, Genetic Drug Design Gene Library High throughput screening (DE-588)4596131-1 gnd Arzneimittelforschung (DE-588)4003120-2 gnd Kombinatorische Synthese (DE-588)4513555-1 gnd |
topic_facet | High throughput screening (Drug development) Combinatorial chemistry Drug development Combinatorial Chemistry Techniques Databases, Genetic Drug Design Gene Library High throughput screening Arzneimittelforschung Kombinatorische Synthese |
url | http://www.loc.gov/catdir/enhancements/fy0829/2007035804-d.html http://www.loc.gov/catdir/toc/fy0804/2007035804.html http://www.gbv.de/dms/bowker/toc/9780849372681.pdf http://bvbr.bib-bvb.de:8991/F?func=service&doc_library=BVB01&local_base=BVB01&doc_number=017597195&sequence=000001&line_number=0001&func_code=DB_RECORDS&service_type=MEDIA |
work_keys_str_mv | AT kshirsagartushar highthroughputleadoptimizationindrugdiscovery |