Strategy in drug research: proceedings of the second IUPAC-IUPHAR Symposium held in Noordwijkerhout (The Netherlands), August 25 - 28, 1981
Saved in:
| Format: | Book |
|---|---|
| Language: | English |
| Published: |
Amsterdam [u.a.]
Elsevier
1982
|
| Series: | Pharmacochemistry library
4 |
| Subjects: | |
| Online Access: | Inhaltsverzeichnis |
| Physical Description: | VIII, 420 S. graph. Darst. |
| ISBN: | 0444420533 |
Staff View
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Record in the Search Index
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| adam_text | IMAGE 1
PHARMACOCHEMISTRY LIBRARY
EDITORS: W.TH. NAUTA AND R.F. REKKER
VOLUME 4
STRATEGY IN DRUG
RESEARCH PROCEEDINGS OF THE SECOND IUPAC-IUPHAR SYMPOSIUM HELD IN
NOORDWIJKERHOUT (THE NETHERLANDS), AUGUST 25-28, 1981 EDITED BY
J.A.KEVERUNGBUISMAN
C/O DUPHAR BV, WEESP, THE NETHERLANDS
ELSEVIER SCIENTIFIC PUBLISHING COMPANY
AMSTERDAM - OXFORD - NEW YORK 1982
IMAGE 2
V
CONTENTS
H. TIMMERMAN PREFACE VII
A.O. LUCAS DRUGS FOR DEVELOPING COUNTRIES 1
H. MOHLER THE BENZODIAZEPINE RECEPTOR AND ITS LIGANDS 13
A. LEVITZKI THE PROBING AND THE MODE OF ACTION OF B- AND A ? -ADRENERGIC
RECEPTORS. . 21 D. ATLAS, M.L. STEER AND Y. PLOTEK CLONIDINE-N=C=S, AN
AFFINITY LABEL FOR A,,-ADRENERGIC RECEPTORS ON
HUMAN PLATELETS AND RAT BRAIN 37
F.J. ZEELEN THE STRATEGY OF THE DEVELOPMENT OF PEPTIDE DRUGS 47
T.A. KRENITSKY AND G.B. EL ION ENZYMES AS TOOLS AND TARGETS IN DRUG
RESEARCH 65
P. BEY, B. METCALF, M.J. JUNG, J. FOZARD AND J. KOCH-WESER
SUBSTRATE-INDUCED IRREVERSIBLE INHIBITION OF ENZYMES IN DRUG RESEARCH .
39 J. KNOLL SELECTIVE INHIBITION OF B TYPE MONOAMINE OXIDASE IN THE
BRAIN: A DRUG
STRATEGY TO IMPROVE THE QUALITY OF LIFE IN SENESCENCE 107
N. BODOR SOFT DRUGS: STRATEGIES FOR DESIGN OF SAFER DRUGS 137
E.J. ARIENS AND A.M. SIMONIS OPTIMALIZATION OF PHARMACOKINETICS -AN
ESSENTIAL ASPECT OF DRUG DEVELOPMENT-BY METABOLIC STABILIZATION 165
J.K. SEYDEL STRUCTURE-PHARMACOKINETICS RELATIONSHIPS IN DRUG DESIGN 179
H. OELSCHLAGER DRUG BIOTRANSFORMATION AS A SOURCE OF DRUG DEVELOPMENT
203
P.J. GOODFORD THE QUANTITATIVE MEASUREMENT OF BIOLOGICAL EFFECTS 223
P.B.M.W.M. TIMMERMANS, A. DE JONGE AND P.A. VAN ZWIETEN QUANTITATIVE
COMPARISONS IN CARDIOVASCULAR PHARMACOLOGY: CHARACTER- IZATION OF
A-ADRENOCEPTOR POPULATIONS 251
Y.C. MARTIN EXAMPLES OF THE ROLE OF COMPUTERS IN NEW COMPOUND DESIGN IN
A PHARMA- CEUTICAL COMPANY 269
A.B. ROZENBLIT COMPUTER-ASSISTED DRUG DESIGN. STRATEGY AND ALGORITHMS
287 E.J. ARIENS STRATEGY IN DRUG RESEARCH - SUMMING UP 309
THE VALUE OF PREDICTIONS IN STRUCTURE-ACTIVITY ANALYSIS : PROCEEDINGS
OF THE SATELLITE SYMPOSIUM QSAR R.F. REKKER THE PREDICTIVE MERITS OF
ANTIHISTAMINE-QSAR STUDIES 315
J.K. SEYDEL AND K.-J. SCHAPER EXCEPTIONS IN QUANTITATIVE
STRUCTURE-ACTIVITY RELATIONSHIPS (QSAR), POSSIBLE REASONS 337
IMAGE 3
VI
R. FRANKE SOME PREREQUISITES AND TECHNIQUES TO MAKE QSARS PREDICTIVE 355
R.M. HYDE AND B. ROTH
SOME ASPECTS OF A QSAR ANALYSIS OF TRIMETHOPRIM ANALOGUES 385
GENERAL (ROUND TABLE) DISCUSSION: PERSPECTIVES IN QSAR 411
LIST OF SYMBOLS USED IN QSAR PUBLICATIONS 413
SUBJECT INDEX 415
|
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| indexdate | 2024-07-09T15:07:50Z |
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| physical | VIII, 420 S. graph. Darst. |
| publishDate | 1982 |
| publishDateSearch | 1982 |
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| series | Pharmacochemistry library |
| series2 | Pharmacochemistry library |
| spelling | Strategy in drug research proceedings of the second IUPAC-IUPHAR Symposium held in Noordwijkerhout (The Netherlands), August 25 - 28, 1981 ed. by J. A. Keverling Buisman Amsterdam [u.a.] Elsevier 1982 VIII, 420 S. graph. Darst. txt rdacontent n rdamedia nc rdacarrier Pharmacochemistry library 4 Pharmazie (DE-588)4045705-9 gnd rswk-swf (DE-588)1071861417 Konferenzschrift 1981 Noordwijkerhout gnd-content Pharmazie (DE-588)4045705-9 s DE-604 Keverling Buisman, Jan A. Sonstige oth International Union of Pure and Applied Chemistry Sonstige (DE-588)1011135-9 oth Pharmacochemistry library 4 (DE-604)BV001899371 4 GBV Datenaustausch application/pdf http://bvbr.bib-bvb.de:8991/F?func=service&doc_library=BVB01&local_base=BVB01&doc_number=000019989&sequence=000001&line_number=0001&func_code=DB_RECORDS&service_type=MEDIA Inhaltsverzeichnis |
| spellingShingle | Strategy in drug research proceedings of the second IUPAC-IUPHAR Symposium held in Noordwijkerhout (The Netherlands), August 25 - 28, 1981 Pharmacochemistry library Pharmazie (DE-588)4045705-9 gnd |
| subject_GND | (DE-588)4045705-9 (DE-588)1071861417 |
| title | Strategy in drug research proceedings of the second IUPAC-IUPHAR Symposium held in Noordwijkerhout (The Netherlands), August 25 - 28, 1981 |
| title_auth | Strategy in drug research proceedings of the second IUPAC-IUPHAR Symposium held in Noordwijkerhout (The Netherlands), August 25 - 28, 1981 |
| title_exact_search | Strategy in drug research proceedings of the second IUPAC-IUPHAR Symposium held in Noordwijkerhout (The Netherlands), August 25 - 28, 1981 |
| title_full | Strategy in drug research proceedings of the second IUPAC-IUPHAR Symposium held in Noordwijkerhout (The Netherlands), August 25 - 28, 1981 ed. by J. A. Keverling Buisman |
| title_fullStr | Strategy in drug research proceedings of the second IUPAC-IUPHAR Symposium held in Noordwijkerhout (The Netherlands), August 25 - 28, 1981 ed. by J. A. Keverling Buisman |
| title_full_unstemmed | Strategy in drug research proceedings of the second IUPAC-IUPHAR Symposium held in Noordwijkerhout (The Netherlands), August 25 - 28, 1981 ed. by J. A. Keverling Buisman |
| title_short | Strategy in drug research |
| title_sort | strategy in drug research proceedings of the second iupac iuphar symposium held in noordwijkerhout the netherlands august 25 28 1981 |
| title_sub | proceedings of the second IUPAC-IUPHAR Symposium held in Noordwijkerhout (The Netherlands), August 25 - 28, 1981 |
| topic | Pharmazie (DE-588)4045705-9 gnd |
| topic_facet | Pharmazie Konferenzschrift 1981 Noordwijkerhout |
| url | http://bvbr.bib-bvb.de:8991/F?func=service&doc_library=BVB01&local_base=BVB01&doc_number=000019989&sequence=000001&line_number=0001&func_code=DB_RECORDS&service_type=MEDIA |
| volume_link | (DE-604)BV001899371 |
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